BENZODIAZEPINE AGONISTS PROTECT A HISTIDINE RESIDUE FROM MODIFICATION BY DIETHYL PYROCARBONATE WHEREAS PROPYL BETA-CARBOLINE DOES NOT

被引：18

作者：

LAMBOLEZ, B

ROSSIER, J

机构：

来源：

FEBS LETTERS | 1987年 / 219卷 / 02期

关键词：

D O I：

10.1016/0014-5793(87)80240-5

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：301 / 305

页数：5

共 12 条

[1] SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].

BRAESTRUP, C ;

SQUIRES, RF .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809

[2]

BURCH TP, 1983, MOL PHARMACOL, V23, P52

[3]

BURCH TP, 1981, P NATL ACAD SCI-BIOL, V78, P3945, DOI 10.1073/pnas.78.6.3945

[4] 3-AMINO-BETA-CARBOLINE DERIVATIVES AND THE BENZODIAZEPINE RECEPTOR - SYNTHESIS OF A SELECTIVE ANTAGONIST OF THE SEDATIVE ACTION OF DIAZEPAM [J].

DODD, RH ;

OUANNES, C ;

DECARVALHO, LP ;

VALIN, A ;

VENAULT, P ;

CHAPOUTHIER, G ;

ROSSIER, J ;

POTIER, P .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (06) :824-828

[5]

Haefely W. E., 1985, ADV DRUG RES, V14, P165

[6]

LOWRY OH, 1951, J BIOL CHEM, V193, P265

[7] CHARACTERIZATION OF GAMMA-AMINOBUTYRIC ACID BENZODIAZEPINE RECEPTOR COMPLEXES BY PROTECTION AGAINST INACTIVATION BY GROUP-SPECIFIC REAGENTS [J].

MAKSAY, G ;

TICKU, MK .

JOURNAL OF NEUROCHEMISTRY, 1984, 42 (06) :1715-1727

[8]

MAUPAS B, 1982, ANALUSIS, V10, P187

[9]

Miles E W, 1977, Methods Enzymol, V47, P431

[10] INVOLVEMENT OF TYROSYL RESIDUES IN THE BINDING OF BENZODIAZEPINES TO THEIR BRAIN RECEPTORS [J].

SHERMANGOLD, R ;

DUDAI, Y .

FEBS LETTERS, 1981, 131 (02) :313-316

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