SYNTHESIS, RECEPTOR-BINDING, AND TISSUE DISTRIBUTION OF (17-ALPHA,20E)-21-[I-125]IODO-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL AND (17-ALPHA,20Z)-21-[I-125]IODO-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL

被引：48

作者：

ALI, H ^{[1
]}

ROUSSEAU, J ^{[1
]}

GHAFFARI, MA ^{[1
]}

VANLIER, JE ^{[1
]}

机构：

[1] UNIV SHERBROOKE,FAC MED,MRC,RADIAT SCI GRP,SHERBROOKE J1H 5N4,QUEBEC,CANADA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 10期

关键词：

D O I：

10.1021/jm00118a013

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1946 / 1950

页数：5

共 12 条

[1]

ALI HDP, UNPUB

[2] THE PREPARATION OF 2 AROMATIC ANALOGS OF DESOXYCORTICOSTERONE ACETATE [J].

DJERASSI, C ;

SCHOLZ, CR .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1949, 71 (12) :3962-3966

[3]

HANSON RN, 1984, J NUCL MED, V25, P998

[4]

HANSON RN, 1982, J NUCL MED, V23, P431

[5] SYNTHESIS OF 17-ALPHA-BROMOVINYLNORTESTOSTERONE AND 17-ALPHA-IODOVINYLNORTESTOSTERONE DERIVATIVES [J].

HOFMEISTER, H ;

LAURENT, H ;

SCHULZE, PE ;

WIECHERT, R .

TETRAHEDRON, 1986, 42 (13) :3575-3578

[6] SYNTHESIS AND EVALUATION OF POTENTIAL RADIOLIGANDS FOR THE PROGESTERONE-RECEPTOR [J].

HOYTE, RM ;

ROSNER, W ;

JOHNSON, IS ;

ZIELINSKI, J ;

HOCHBERG, RB .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (11) :1695-1699

[7] Testings on sex hormone array [J].

Inhoffen, HH ;

Logemann, W ;

Hohlweg, W ;

Serini, A .

BERICHTE DER DEUTSCHEN CHEMISCHEN GESELLSCHAFT, 1938, 71 :1024-1032

[8]

JAGODA EM, 1984, J NUCL MED, V25, P472

[9]

KIRSCHNER AS, 1975, J NUCL MED, V16, P248

[10] SYNTHESIS AND EVALUATION OF (17-ALPHA,20E)-21-[I-125]IODO-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL AND (17-ALPHA,20E)-21-[I-125]IODO-11-BETA-METHOXY-19-NORPREGNA-1,3,5(10),20-TETRAENE-3,17-DIOL (17-ALPHA-(IODOVINYL)ESTRADIOL DERIVATIVES) AS HIGH SPECIFIC ACTIVITY POTENTIAL RADIOPHARMACEUTICALS-1 [J].

NAKATSUKA, I ;

FERREIRA, NL ;

ECKELMAN, WC ;

FRANCIS, BE ;

RZESZOTARSKI, WJ ;

GIBSON, RE ;

JAGODA, EM ;

REBA, RC .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (10) :1287-1291

← 1 2 →