CLINICAL-PHARMACOLOGY OF TRIMETREXATE

被引:17
作者
HO, DHW
COVINGTON, WP
LEGHA, SS
NEWMAN, RA
KRAKOFF, IH
机构
关键词
D O I
10.1038/clpt.1987.160
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:351 / 356
页数:6
相关论文
共 24 条
[1]  
BALIS FM, 1986, CANCER RES, V46, P169
[2]  
BALIS FM, 1985, P AM SOC CLIN ONCOL, V4, P35
[3]   ESTRIP, A BASIC COMPUTER-PROGRAM FOR OBTAINING INITIAL POLYEXPONENTIAL PARAMETER ESTIMATES [J].
BROWN, RD ;
MANNO, JE .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1978, 67 (12) :1687-1691
[4]  
DIDDENS H, 1983, CANCER RES, V43, P5286
[5]   DRUG METABOLISM AFTER REPEATED TREATMENTS WITH CYTOTOXIC AGENTS [J].
DONELLI, MG ;
GARATTINI, S .
EUROPEAN JOURNAL OF CANCER, 1971, 7 (04) :361-+
[6]  
GIBALDI M, 1974, PHARMACOKINETICS, P281
[7]   ENZYMATIC ASSAYS FOR 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL]QUINAZOLINE, A PROMISING NEW NON-CLASSICAL ANTIFOLATE [J].
HEUSNER, JJ ;
MCCORMACK, JJ .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (07) :827-828
[8]  
HEUSNER JJ, 1985, P AM ASSOC CANC RES, V26, P234
[9]   BIOCHEMICAL PHARMACOLOGY OF THE LIPOPHILIC ANTIFOLATE, TRIMETREXATE [J].
JACKSON, RC ;
FRY, DW ;
BORITZKI, TJ ;
BESSERER, JA ;
LEOPOLD, WR ;
SLOAN, BJ ;
ELSLAGER, EF .
ADVANCES IN ENZYME REGULATION, 1984, 22 :187-206
[10]   UPTAKE AND EFFICACY OF TRIMETREXATE (TMQ, 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL] QUINAZOLINE), A NON-CLASSICAL ANTIFOLATE IN METHOTREXATE-RESISTANT LEUKEMIA-CELLS INVITRO [J].
KAMEN, BA ;
EIBL, B ;
CASHMORE, A ;
BERTINO, J .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (10) :1697-1699