SCREENING OF ANTI-PROGESTAGENS BY RECEPTOR STUDIES AND BIOASSAYS

被引：37

作者：

KLOOSTERBOER, HJ ^{[1
]}

DECKERS, GHJ ^{[1
]}

VANDERHEUVEL, MJ ^{[1
]}

LOOZEN, HJJ ^{[1
]}

机构：

[1] ORGANON SCI DEV GRP, OSS, NETHERLANDS

来源：

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY | 1988年 / 31卷 / 4B期

关键词：

D O I：

10.1016/0022-4731(88)90007-6

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：567 / 571

页数：5

共 14 条

[1] RU486, A PROGESTIN AND GLUCOCORTICOID ANTAGONIST, INHIBITS THE GROWTH OF BREAST-CANCER CELLS VIA THE PROGESTERONE-RECEPTOR [J].

BARDON, S ;

VIGNON, F ;

CHALBOS, D ;

ROCHEFORT, H .

JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1985, 60 (04) :692-697

[2] REGIO AND STEREOSPECIFIC SYNTHESIS OF 11-BETA-SUBSTITUTED 19-NORSTEROIDS - INFLUENCE OF 11-BETA-SUBSTITUTION ON PROGESTERONE-RECEPTOR AFFINITY [J].

BELANGER, A ;

PHILIBERT, D ;

TEUTSCH, G .

STEROIDS, 1981, 37 (04) :361-382

[3] BINDING OF PROGESTAGENS TO RECEPTOR PROTEINS IN MCF-7 CELLS [J].

BERGINK, EW ;

VANMEEL, F ;

TURPIJN, EW ;

VANDERVIES, J .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1983, 19 (05) :1563-1570

[4] PROGESTERONE-RECEPTOR BLOCKAGE - EFFECT ON UTERINE CONTRACTILITY AND EARLY-PREGNANCY [J].

BYGDEMAN, M ;

SWAHN, ML .

CONTRACEPTION, 1985, 32 (01) :45-51

[5]

ELGER W, 1985, Journal of Steroid Biochemistry, V23, p11S

[6]

HERRMANN W, 1982, CR ACAD SCI III-VIE, V294, P933

[7] TERMINATION OF VERY EARLY-PREGNANCY BY RU-486 - AN ANTIPROGESTATIONAL COMPOUND [J].

KOVACS, L ;

SAS, M ;

RESCH, BA ;

UGOCSAI, G ;

SWAHN, ML ;

BYGDEMAN, M ;

ROWE, PJ .

CONTRACEPTION, 1984, 29 (05) :399-410

[8] SUCCESSFUL TREATMENT OF CUSHINGS-SYNDROME WITH THE GLUCOCORTICOID ANTAGONIST RU-486 [J].

NIEMAN, LK ;

CHROUSOS, GP ;

KELLNER, C ;

SPITZ, IM ;

NISULA, BC ;

CUTLER, GB ;

MERRIAM, GR ;

BARDIN, CW ;

LORIAUX, DL .

JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1985, 61 (03) :536-540

[9] A NEW SUBSTANCE WITH PROGESTATIONAL ACTIVITY .2. PHARMACOLOGICAL PROPERTIES [J].

OVERBEEK, GA ;

DEVISSER, J .

ACTA ENDOCRINOLOGICA, 1956, 22 (04) :318-329

[10]

PHILIBERT D, 1982, RU 38486 NEW LEAD ST

← 1 2 →