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THE EFFECT OF NMETYR(5) SUBSTITUTION IN LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONISTS
被引:25
作者
:
HAVIV, F
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
HAVIV, F
[
1
]
FITZPATRICK, TD
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
FITZPATRICK, TD
[
1
]
NICHOLS, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
NICHOLS, CJ
[
1
]
SWENSON, RE
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
SWENSON, RE
[
1
]
MORT, NA
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
MORT, NA
[
1
]
BUSH, EN
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
BUSH, EN
[
1
]
DIAZ, G
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
DIAZ, G
[
1
]
NGUYEN, AT
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
NGUYEN, AT
[
1
]
HOLST, MR
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
HOLST, MR
[
1
]
CYBULSKI, VA
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
CYBULSKI, VA
[
1
]
LEAL, JA
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
LEAL, JA
[
1
]
BAMMERT, G
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
BAMMERT, G
[
1
]
RHUTASEL, NS
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
RHUTASEL, NS
[
1
]
DODGE, PW
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
DODGE, PW
[
1
]
JOHNSON, ES
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
JOHNSON, ES
[
1
]
CANNON, JB
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
CANNON, JB
[
1
]
KNITTLE, J
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
KNITTLE, J
[
1
]
GREER, J
论文数:
0
引用数:
0
h-index:
0
机构:
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
GREER, J
[
1
]
机构
:
[1]
ABBOTT LABS, DIV PROD, ABBOTT PK, IL 60064 USA
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1993年
/ 36卷
/ 07期
关键词
:
D O I
:
10.1021/jm00059a020
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:928 / 933
页数:6
相关论文
共 35 条
[1]
HIGHLY POTENT ANTAGONISTS OF LUTEINIZING-HORMONE-RELEASING HORMONE FREE OF EDEMATOGENIC EFFECTS
BAJUSZ, S
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
BAJUSZ, S
KOVACS, M
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
KOVACS, M
GAZDAG, M
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
GAZDAG, M
BOKSER, L
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
BOKSER, L
KARASHIMA, T
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
KARASHIMA, T
CSERNUS, VJ
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
CSERNUS, VJ
JANAKY, T
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
JANAKY, T
GUOTH, J
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
GUOTH, J
SCHALLY, AV
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
SCHALLY, AV
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1988,
85
(05)
: 1637
-
1641
[2]
NUCLEAR-MAGNETIC-RESONANCE ANALYSIS AND CONFORMATIONAL CHARACTERIZATION OF A CYCLIC DECAPEPTIDE ANTAGONIST OF GONADOTROPIN-RELEASING-HORMONE
BANIAK, EL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
BANIAK, EL
RIVIER, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
RIVIER, JE
STRUTHERS, RS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
STRUTHERS, RS
HAGLER, AT
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
HAGLER, AT
GIERASCH, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
GIERASCH, LM
[J].
BIOCHEMISTRY,
1987,
26
(09)
: 2642
-
2656
[3]
PROLONGED INHIBITION OF LUTEINIZING-HORMONE AND TESTOSTERONE LEVELS IN MALE-RATS WITH THE LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONIST SB-75
BOKSER, L
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
BOKSER, L
BAJUSZ, S
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
BAJUSZ, S
GROOT, K
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
GROOT, K
SCHALLY, AV
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
SCHALLY, AV
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1990,
87
(18)
: 7100
-
7104
[4]
BUSH EN, 1992, 74TH ANN M END SOC S
[5]
BUSH EN, UNPUB ENDOCRINOLOGY
[6]
CHAN RL, 1991, DRUG METAB DISPOS, V19, P858
[7]
DECKERS GHJ, 1989, 71ST ANN M END SOC S
[8]
DUTTA A S, 1988, Drugs of the Future, V13, P43
[9]
SINGLE DOSE LONG-TERM SUPPRESSION OF TESTOSTERONE SECRETION BY A GONADOTROPIN-RELEASING-HORMONE ANTAGONIST (ANTIDE) IN MALE MONKEYS
EDELSTEIN, MC
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EDELSTEIN, MC
GORDON, K
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
GORDON, K
WILLIAMS, RF
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
WILLIAMS, RF
DANFORTH, DR
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
DANFORTH, DR
HODGEN, GD
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
HODGEN, GD
[J].
CONTRACEPTION,
1990,
42
(02)
: 209
-
214
[10]
GNRH AGONISTS AND ANTAGONISTS - CURRENT CLINICAL STATUS
FILICORI, M
论文数:
0
引用数:
0
h-index:
0
FILICORI, M
FLAMIGNI, C
论文数:
0
引用数:
0
h-index:
0
FLAMIGNI, C
[J].
DRUGS,
1988,
35
(01)
: 63
-
82
←
1
2
3
4
→
共 35 条
[1]
HIGHLY POTENT ANTAGONISTS OF LUTEINIZING-HORMONE-RELEASING HORMONE FREE OF EDEMATOGENIC EFFECTS
BAJUSZ, S
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
BAJUSZ, S
KOVACS, M
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
KOVACS, M
GAZDAG, M
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
GAZDAG, M
BOKSER, L
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
BOKSER, L
KARASHIMA, T
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
KARASHIMA, T
CSERNUS, VJ
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
CSERNUS, VJ
JANAKY, T
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
JANAKY, T
GUOTH, J
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
GUOTH, J
SCHALLY, AV
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
TULANE UNIV,SCH MED,DEPT MED,NEW ORLEANS,LA 70146
SCHALLY, AV
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1988,
85
(05)
: 1637
-
1641
[2]
NUCLEAR-MAGNETIC-RESONANCE ANALYSIS AND CONFORMATIONAL CHARACTERIZATION OF A CYCLIC DECAPEPTIDE ANTAGONIST OF GONADOTROPIN-RELEASING-HORMONE
BANIAK, EL
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
BANIAK, EL
RIVIER, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
RIVIER, JE
STRUTHERS, RS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
STRUTHERS, RS
HAGLER, AT
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
HAGLER, AT
GIERASCH, LM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV DELAWARE,DEPT CHEM,NEWARK,DE 19716
GIERASCH, LM
[J].
BIOCHEMISTRY,
1987,
26
(09)
: 2642
-
2656
[3]
PROLONGED INHIBITION OF LUTEINIZING-HORMONE AND TESTOSTERONE LEVELS IN MALE-RATS WITH THE LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONIST SB-75
BOKSER, L
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
BOKSER, L
BAJUSZ, S
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
BAJUSZ, S
GROOT, K
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
GROOT, K
SCHALLY, AV
论文数:
0
引用数:
0
h-index:
0
机构:
TULANE UNIV,VET ADM MED CTR,SCH MED,NEW ORLEANS,LA 70146
SCHALLY, AV
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1990,
87
(18)
: 7100
-
7104
[4]
BUSH EN, 1992, 74TH ANN M END SOC S
[5]
BUSH EN, UNPUB ENDOCRINOLOGY
[6]
CHAN RL, 1991, DRUG METAB DISPOS, V19, P858
[7]
DECKERS GHJ, 1989, 71ST ANN M END SOC S
[8]
DUTTA A S, 1988, Drugs of the Future, V13, P43
[9]
SINGLE DOSE LONG-TERM SUPPRESSION OF TESTOSTERONE SECRETION BY A GONADOTROPIN-RELEASING-HORMONE ANTAGONIST (ANTIDE) IN MALE MONKEYS
EDELSTEIN, MC
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EDELSTEIN, MC
GORDON, K
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
GORDON, K
WILLIAMS, RF
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
WILLIAMS, RF
DANFORTH, DR
论文数:
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引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
DANFORTH, DR
HODGEN, GD
论文数:
0
引用数:
0
h-index:
0
机构:
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
EASTERN VIRGINIA MED SCH,JONES INST REPROD MED,DEPT OBSTET & GYNECOL,NORFOLK,VA 23510
HODGEN, GD
[J].
CONTRACEPTION,
1990,
42
(02)
: 209
-
214
[10]
GNRH AGONISTS AND ANTAGONISTS - CURRENT CLINICAL STATUS
FILICORI, M
论文数:
0
引用数:
0
h-index:
0
FILICORI, M
FLAMIGNI, C
论文数:
0
引用数:
0
h-index:
0
FLAMIGNI, C
[J].
DRUGS,
1988,
35
(01)
: 63
-
82
←
1
2
3
4
→