A FACILE AND EFFICIENT METHOD FOR MACROLACTAMIZATION

被引：6

作者：

BAI, DL

BO, YX

ZHOU, QT

机构：

[1] Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 15期

关键词：

D O I：

10.1016/0040-4039(90)80098-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Using 2-bromo-l-methylpyridinium iodide as carboxyl activating agent, 10 ansa-macrolactams were prepared conveniently from the corresponding seco-precursor ω-amino acids. In most cases the yields are excellent. © 1990.

引用

页码：2161 / 2164

页数：4

共 9 条

[1] FACILE SYNTHESIS OF CARBOXAMIDES BY USING 1-METHYL-2-HALOPYRIDINIUM IODIDES AS COUPLING REAGENTS [J].

BALD, E ;

SAIGO, K ;

MUKAIYAMA, T .

CHEMISTRY LETTERS, 1975, (11) :1163-1166

[2] TOTAL SYNTHESIS OF MAYTANSINE [J].

COREY, EJ ;

WEIGEL, LO ;

CHAMBERLIN, AR ;

CHO, H ;

HUA, DH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (21) :6613-6615

[3]

GU XQ, 1988, SCI CHINA SER B, V31, P1342

[4] TOTAL SYNTHESIS OF RIFAMYCINS .2. TOTAL SYNTHESIS OF RACEMIC RIFAMYCIN-S [J].

IIO, H ;

NAGAOKA, H ;

KISHI, Y .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (27) :7965-7967

[5]

MARCH J, 1985, ADV ORGANIC CHEM

[6] FACILE SYNTHESIS OF LACTONES [J].

MUKAIYAMA, T ;

USUI, M ;

SAIGO, K .

CHEMISTRY LETTERS, 1976, (01) :49-50

[7] NOVEL SYNTHESIS OF OMEGA-(DIPHENYLPHOSPHINYL)ALKYLCARBOXYLIC ACIDS FROM TRIPHENYL-OMEGA-CARBOXYALKYLPHOSPHONIUM SALTS [J].

NARAYANAN, KS ;

BERLIN, KD .

JOURNAL OF ORGANIC CHEMISTRY, 1980, 45 (11) :2240-2243

[8] RECENT DEVELOPMENTS IN THE TOTAL SYNTHESIS OF MACROLIDE ANTIBIOTICS [J].

PATERSON, I ;

MANSURI, MM .

TETRAHEDRON, 1985, 41 (18) :3569-3624

[9]

ZHOU QT, 1986, KEXUE TONGBAO, V31, P806

← 1 →