PYRIMIDO[4,5-C]PYRIDAZINES .3. PREFERENTIAL FORMATION OF 8-AMINO-1H-PYRIMIDO[4,5-C]-1,2-DIAZEPIN-6(7H)-ONES BY CYCLIZATIONS WITH ALPHA,GAMMA-DIKETO ESTERS

被引：18

作者：

MALLORY, WR ^{[1
]}

MORRISON, RW ^{[1
]}

STYLES, VL ^{[1
]}

机构：

[1] BURROUGHS WELLCOME CO,WELLCOME RES LABS,RES TRIANGLE PK,NC 27709

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1982年 / 47卷 / 04期

关键词：

D O I：

10.1021/jo00343a013

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：667 / 674

页数：8

共 12 条

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KLINGSBE.E .

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[6]

LAIRD AH, 1961, Patent No. 876601

[7] PYRIMIDO[4,5-C]PYRIDAZINES .1. CYCLIZATIONS WITH ALPHA-KETO ESTERS [J].

MORRISON, RW ;

MALLORY, WR ;

STYLES, VL .

JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (25) :4844-4849

[8] CHEMISTRY OF 1,2-DIAZEPINES [J].

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[9]

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[10]

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