A NOVEL IMIDAZOLIDIN-2-ONE AUXILIARY FOR A HIGHLY STEREOSELECTIVE ALDOL ROUTE TO BETA-HYDROXYESTERS

被引：13

作者：

DREWES, SE ^{[1
]}

MALISSAR, DGS ^{[1
]}

ROOS, GHP ^{[1
]}

机构：

[1] UNIV NATAL,DEPT CHEM,BOX 375,PIETERMARITZBURG 3200,SOUTH AFRICA

来源：

TETRAHEDRON-ASYMMETRY | 1992年 / 3卷 / 04期

关键词：

D O I：

10.1016/S0957-4166(00)80254-2

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Enantiomerically pure syn-aldols are obtained from the boron enolate of (4R, 5S)-1,5-dimethyl-4-cyclohexyl-3- propanoyl imidazolidin-2-one. Cleavage of the auxiliary affords the homochiral title esters in good yield.

引用

页码：515 / 516

页数：2

共 8 条

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