IMPORTANCE OF THE N-TERMINAL DOMAIN OF THE TYPE-II ANGIOTENSIN ANTAGONIST SARMESIN FOR RECEPTOR BLOCKADE

被引：38

作者：

MATSOUKAS, J

CORDOPATIS, P

BELTE, U

GOGHARI, MH

GANTER, RC

FRANKLIN, KJ

MOORE, GJ

机构：

[1] UNIV CALGARY,DEPT MED BIOCHEM,CALGARY T2N 4N1,ALBERTA,CANADA

[2] UNIV PATRAS,DEPT CHEM,PATRAS,GREECE

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 07期

关键词：

D O I：

10.1021/jm00402a028

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1418 / 1421

页数：4

共 11 条

[1]

FERMANDJIAN S, 1976, PEPTIDES 1976, P339

[2] STRUCTURE-ACTIVITY-RELATIONSHIPS FOR THE COMPETITIVE ANGIOTENSIN ANTAGONIST [SARCOSINE1,O-METHYLTYROSINE4]ANGIOTENSIN-II (SARMESIN) [J].

GOGHARI, MH ;

FRANKLIN, KJ ;

MOORE, GJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (06) :1121-1124

[3] PROTON MAGNETIC-RESONANCE STUDIES OF ANGIOTENSIN-II CONFORMATION - CIS-TRANS ISOMERISM IN SARCOSINE-7-CONTAINING ANALOGS [J].

MATSOUKAS, JM ;

MOORE, GJ .

ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1986, 248 (01) :419-423

[4] SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF ANALOGS OF ANGIOTENSIN-II AND ANGIOTENSIN-III CONTAINING O-METHYLTYROSINE AND D-TRYPTOPHAN [J].

MATSOUKAS, JM ;

GOGHARI, MH ;

SCANLON, MN ;

FRANKLIN, KJ ;

MOORE, GJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (06) :780-783

[5] STRUCTURE DESENSITIZATION RELATIONSHIPS OF ANGIOTENSIN ANALOGS IN THE RAT ISOLATED UTERUS [J].

MOORE, GJ ;

FRANKLIN, KJ ;

NYSTROM, DM ;

GOGHARI, MH .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1985, 63 (08) :966-971

[6]

MOORE GJ, 1985, INT J PEPT PROT RES, V26, P469

[7]

MOORE GJ, 1985, BIOSCIENCE REP, V58, P407

[8] A NEW APPROACH TO ANGIOTENSIN ANTAGONISTS - METHYLATION OF THE TYROSINE HYDROXYL IN ANGIOTENSIN-II [J].

SCANLON, MN ;

MATSOUKAS, JM ;

FRANKLIN, KJ ;

MOORE, GJ .

LIFE SCIENCES, 1984, 34 (04) :317-321

[9]

SMEBY RR, 1978, CHEM BIOCH AMINO ACI, V5, P117

[10] NEW, LONG-LASTING COMPETITIVE INHIBITOR OF ANGIOTENSIN [J].

TURKER, RK ;

SWEET, CS ;

YAMAMOTO, M ;

BUMPUS, FM ;

HALL, MM .

SCIENCE, 1972, 177 (4055) :1203-&

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