METHOXYLATION OF COCAINE REDUCES BINDING-AFFINITY AND PRODUCES COMPOUNDS OF DIFFERENTIAL BINDING AND DOPAMINE UPTAKE INHIBITORY ACTIVITY - DISCOVERY OF A WEAK COCAINE ANTAGONIST

被引：66

作者：

SIMONI, D

STOELWINDER, J

KOZIKOWSKI, AP

JOHNSON, KM

BERGMANN, JS

BALL, RG

机构：

[1] MAYO FDN MED EDUC & RES,JACKSONVILLE,FL 32224

[2] UNIV TEXAS,MED BRANCH,DEPT PHARMACOL & TOXICOL,GALVESTON,TX 77555

[3] MERCK SHARP & DOHME LTD,RES LABS,RAHWAY,NJ 07065

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1993年 / 36卷 / 24期

关键词：

D O I：

10.1021/jm00076a028

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：3975 / 3977

页数：3

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