A SIMPLE GENERAL-METHOD FOR (RADIO)IODINATION OF A PHENYLALANINE RESIDUE IN PEPTIDES - PREPARATION OF [D-PEN(2),4'-I-125-PHE(4),D-PEN(5)]ENKEPHALIN, A PEPTIDE WITH EXTRAORDINARY SELECTIVITY FOR DELTA-OPIOID RECEPTORS

被引：18

作者：

SHARMA, SD ^{[1
]}

TOTH, G ^{[1
]}

HRUBY, VJ ^{[1
]}

机构：

[1] UNIV ARIZONA, DEPT CHEM, TUCSON, AZ 85721 USA

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1991年 / 56卷 / 16期

关键词：

D O I：

10.1021/jo00016a035

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：4981 / 4983

页数：3

共 18 条

[1]

Bolton A E, 1986, Methods Enzymol, V124, P18

[2] (S)-N-[(1-ETHYL-2-PYRROLIDINYL)METHYL]-5-[I-125]IODO-2-METHOXYBENZAMIDE HYDROCHLORIDE, A NEW SELECTIVE RADIOLIGAND FOR DOPAMINE D-2 RECEPTORS [J].

DEPAULIS, T ;

JANOWSKY, A ;

KESSLER, RM ;

CLANTON, JA ;

SMITH, HE .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (10) :2027-2033

[3] A NEW METHOD OF IODINE LABELING OF PEPTIDE-HORMONES [J].

ESCHER, E .

JOURNAL OF RECEPTOR RESEARCH, 1984, 4 (1-6) :331-336

[4]

Hartwell JL, 1944, ORG SYNTH, V24, P22

[5] PROSTHETIC GROUP RADIOIODINATION AT NO-CARRIER ADDED LEVELS OF CARBONYL-CONTAINING MOLECULES [J].

HEINDEL, ND ;

VANDORT, M .

JOURNAL OF ORGANIC CHEMISTRY, 1985, 50 (11) :1988-1990

[6] EFFECTS OF CHLORAMINE T AND IODINATION ON THE BIOLOGICAL-ACTIVITY OF MELANOTROPIN [J].

HEWARD, CB ;

YANG, YCS ;

ORMBERG, JF ;

HADLEY, ME ;

HRUBY, VJ .

HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1979, 360 (12) :1851-1859

[7] RECENT DEVELOPMENTS IN THE DESIGN OF RECEPTOR SPECIFIC OPIOID-PEPTIDES [J].

HRUBY, VJ ;

GEHRIG, CA .

MEDICINAL RESEARCH REVIEWS, 1989, 9 (03) :343-401

[8]

KNAPP RJ, 1990, ADV PAIN RES THER, V14, P45

[9]

KNAPP RJ, IN PRESS J PHARM EXP

[10] SYNTHESIS OF HIGHLY MU-OPIOID AND DELTA-OPIOID RECEPTOR SELECTIVE PEPTIDES CONTAINING A PHOTOAFFINITY GROUP [J].

LANDIS, G ;

LUI, G ;

SHOOK, JE ;

YAMAMURA, HI ;

BURKS, TF ;

HRUBY, VJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (03) :638-643

← 1 2 →