C-2-SYMMETRICAL PHOSPHINIC ACID INHIBITORS OF HIV PROTEASE

被引：106

作者：

PEYMAN, A

BUDT, KH

SPANIG, J

STOWASSER, B

RUPPERT, D

机构：

[1] Hoechst AG, Pharma Forschung G838

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 32期

关键词：

D O I：

10.1016/S0040-4039(00)61309-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of the previously not accessible symmetrical bis(alpha-aminoalkyl)phosphinic acids is demonstrated. These compounds are valuable central building blocks in the synthesis of HIV protease inhibitors.

引用

页码：4549 / 4552

页数：4

共 26 条

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