SPINAL ACTIONS OF SUBSTANCE P-ANALOGS ON CARDIOVASCULAR-RESPONSES IN THE RAT - A STRUCTURE ACTIVITY ANALYSIS

被引:9
作者
COUTURE, R [1 ]
GUPTA, A [1 ]
KEROUAC, R [1 ]
ESCHER, E [1 ]
REGOLI, D [1 ]
机构
[1] UNIV SHERBROOKE, FAC MED, DEPT PHYSIOL & PHARMACOL, SHERBROOKE J1H 5N4, QUEBEC, CANADA
关键词
D O I
10.1139/y87-069
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:412 / 418
页数:7
相关论文
共 26 条
  • [1] INTRATHECAL (D-PRO2,D-TRP7,9)-SP ELICITS HYPOALGESIA AND MOTOR BLOCKADE IN THE RAT AND ANTAGONIZES NOXIOUS RESPONSES INDUCED BY SUBSTANCE-P
    AKERMAN, B
    ROSELL, S
    FOLKERS, K
    [J]. ACTA PHYSIOLOGICA SCANDINAVICA, 1982, 114 (04): : 631 - 633
  • [2] SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF SUBSTANCE-P ANTAGONISTS
    CARANIKAS, S
    MIZRAHI, J
    ESCHER, E
    REGOLI, D
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (11) : 1313 - 1316
  • [3] CHARACTERIZATION OF SPINAL ACTIONS OF 4 SUBSTANCE-P ANALOGS
    COUTURE, R
    YASHPAL, K
    HENRY, JL
    ESCHER, E
    REGOLI, D
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 110 (01) : 63 - 69
  • [4] COUTURE R, 1987, IN PRESS J CARDIOVAS
  • [5] COUTURE R, 1987, IN PRESS EUR J PHARM
  • [6] NEW TABLES FOR MULTIPLE COMPARISONS WITH CONTROL
    DUNNETT, CW
    [J]. BIOMETRICS, 1964, 20 (03) : 482 - &
  • [7] A SUBSTANCE-P ANTAGONIST NOT CONTAINING D-TRYPTOPHAN
    ESCHER, E
    DORLEANSJUSTE, P
    DION, S
    DRAPEAU, G
    MIZRAHI, J
    REGOLI, D
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 105 (3-4) : 375 - 377
  • [8] DESIGN AND SYNTHESIS OF EFFECTIVE ANTAGONISTS OF SUBSTANCE-P
    FOLKERS, K
    HORIG, J
    RAMPOLD, G
    LANE, P
    ROSELL, S
    BJORKROTH, U
    [J]. ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1982, 36 (06): : 389 - 395
  • [9] A SUBSTANCE-P ANTAGONIST, [D-PRO2, D-TRP7,9]SP, INHIBITS INFLAMMATORY RESPONSES IN THE RABBIT EYE
    HOLMDAHL, G
    HAKANSON, R
    LEANDER, S
    ROSELL, S
    FOLKERS, K
    SUNDLER, F
    [J]. SCIENCE, 1981, 214 (4524) : 1029 - 1031
  • [10] JONES RSG, 1983, SUBSTANCE P, P237