SYNTHESIS AND BIOCHEMICAL EVALUATION OF INHIBITORS OF ESTROGEN BIOSYNTHESIS

被引：93

作者：

BRUEGGEMEIER, RW

FLOYD, EE

COUNSELL, RE

机构：

[1] UNIV MICHIGAN,DEPT PHARMACOL,ANN ARBOR,MI 48109

[2] UNIV MICHIGAN,INTERDEPT PROGRAM MED CHEM,ANN ARBOR,MI 48109

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1978年 / 21卷 / 10期

关键词：

D O I：

10.1021/jm00208a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1007 / 1011

页数：5

共 27 条

[1] ACTIVE-SITE-DIRECTED INACTIVATION OF AROMATASE FROM HUMAN PLACENTAL MICROSOMES BY BROMINATED ANDROGEN DERIVATIVES
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[2] CYTOTOXIC COMPOUNDS .1. PARA-(NN-DI-2'-CHLOROETHYL-AMINO)THIOPHENOL AND PARA-(NN-DI-2'-BROMOETHYL-AMINO)THIOPHENOL
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OWEN, LN
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[J]. JOURNAL OF THE CHEMICAL SOCIETY, 1958, (AUG): : 2800 - 2810
[3] BRUEGGEMEIER R, 1977, 174TH NAT M AM CHEM
[4] BRUEGGEMEIER RW, 1977, THESIS U MICHIGAN
[5] THE DIRECT CONVERSION OF STEROIDAL DELTA-5-3-BETA-ALCOHOLS TO DELTA-5-KETONES AND DELTA-4-3-KETONES
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[J]. JOURNAL OF ORGANIC CHEMISTRY, 1956, 21 (12) : 1547 - 1548
[6] ADDITION OF ALKANETHIOLIC ACIDS TO DELTA-1,4-3-OXO- AND DELTA-4,6-3-OXOSTEROIDS
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[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1959, 81 (05) : 1224 - 1227
[7] THE PREPARATION OF MERCAPTANS FROM ALCOHOLS
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[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1946, 68 (10) : 2103 - 2104
[8] PARTICIPATION OF A NONENZYMATIC TRANSFORMATION IN BIOSYNTHESIS OF ESTROGENS FROM ANDROGENS
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[J]. SCIENCE, 1977, 195 (4273) : 80 - 81
[9] ANTI-PROGESTATIONAL AGENTS - SYNTHESIS OF 7-ALKYL STEROIDAL KETONES WITH ANTI-IMPLANTATIONAL AND ANTI-DECIDUAL ACTIVITY
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JOHNSTON, JO
PETROW, V
[J]. STEROIDS, 1976, 27 (06) : 759 - 771
[10] BIOSYNTHESIS OF ESTROGENS
GUAL, C
GUT, M
MORATO, T
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HAYANO, M
[J]. ENDOCRINOLOGY, 1962, 71 (06) : 920 - &

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