SYNTHESIS AND CCK-B BINDING AFFINITIES OF CYCLIC ANALOGS OF THE POTENT AND SELECTIVE CCK-B RECEPTOR ANTAGONIST CIL-988

被引：15

作者：

DIDIER, E ^{[1
]}

HORWELL, DC ^{[1
]}

PRITCHARD, MC ^{[1
]}

机构：

[1] PARKE DAVIS & CO, NEUROSCI RES CTR, ADDENBROOKES HOSP SITE, HILLS RD, CAMBRIDGE CB2 2QB, ENGLAND

来源：

TETRAHEDRON | 1992年 / 48卷 / 39期

关键词：

D O I：

10.1016/S0040-4020(01)86596-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A selected series of 14-membered macrocyclic compounds (2) has been prepared as potential CCK-B receptor selective ligands. The efficiency of a number of cyclising reagents has also been evaluated.

引用

页码：8471 / 8490

页数：20

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