A SHORT SYNTHESIS OF A BIPHENOMYCIN-B ANALOG VIA A DOUBLE HECK COUPLING PROCEDURE

被引：20

作者：

CARLSTROM, AS ^{[1
]}

FREJD, T ^{[1
]}

机构：

[1] LUND INST TECHNOL,CTR CHEM,S-22100 LUND,SWEDEN

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1991年 / 17期

关键词：

D O I：

10.1039/c39910001216

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A biphenomycin B analogue has been prepared using the double Heck coupling of 3,3'-diiodo-4,4'-dimethoxybiphenyl and two orthogonally protected 2-amidoacrylates followed by two peptide bond forming steps for the incorporation of L-lysine as the middle amino acid residue.

引用

页码：1216 / 1217

页数：2

共 19 条

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