EVIDENCE FOR THE EXISTENCE OF AT LEAST 2 DIFFERENT BINDING-SITES FOR 5HT-REUPTAKE INHIBITORS WITHIN THE 5HT-REUPTAKE SYSTEM FROM HUMAN-PLATELETS

被引:32
作者
BIESSEN, EAL [1 ]
NORDER, JA [1 ]
HORN, AS [1 ]
ROBILLARD, GT [1 ]
机构
[1] UNIV GRONINGEN,DEPT PHYS CHEM,9713 AW GRONINGEN,NETHERLANDS
关键词
D O I
10.1016/0006-2952(88)90080-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3959 / 3966
页数:8
相关论文
共 19 条
[1]  
ADLER H, 1986, EUR J PHARM, V116, P175
[2]   SELECTIVE EFFECTS OF THIOL REAGENTS ON THE BINDING-SITES FOR IMIPRAMINE AND NEUROTRANSMITTER AMINES IN THE RAT-BRAIN [J].
BIASSONI, R ;
VACCARI, A .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 85 (02) :447-456
[3]   TEMPERATURE-SENSITIVE CONFORMATIONAL-CHANGES IN [H-3]IMIPRAMINE BINDING-SITES AND THE INVOLVEMENT OF SULFUR-CONTAINING BONDS [J].
DAVIS, A .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 102 (02) :341-347
[4]   MOLECULAR ASPECTS OF THE IMIPRAMINE RECEPTOR [J].
DAVIS, A .
EXPERIENTIA, 1984, 40 (08) :782-794
[5]  
FREEDMAN RB, 1978, TECHNIQUES PROTEIN E, V117, P1
[6]  
KEIGHTLEY DD, 1980, J STER BIOCH, V13, P1312
[7]   DOPAMINE RECEPTOR TURNOVER RATES IN RAT STRIATUM ARE AGE-DEPENDENT [J].
LEFF, SE ;
GARIANO, R ;
CREESE, I .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (12) :3910-3914
[8]  
MELLER E, 1985, J PHARMACOL EXP THER, V233, P656
[9]   HIGH-AFFINITY BINDING OF [H-3]LABELED PAROXETINE AND [H-3]IMIPRAMINE TO HUMAN-PLATELET MEMBRANES [J].
MELLERUP, ET ;
PLENGE, P ;
ENGELSTOFT, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 96 (3-4) :303-309
[10]   SIZE DETERMINATION OF BINDING POLYMERS FOR [H-3]IMIPRAMINE AND [H-3] PAROXETINE IN HUMAN-PLATELET MEMBRANES [J].
MELLERUP, ET ;
PLENGE, P ;
NIELSEN, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 106 (02) :411-413