SYNTHESIS, BINDING-STUDIES, AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 1-ARYL[1]BENZOPYRANOPYRAZOL-4-ONES AND 2-ARYL[1]BENZOPYRANOPYRAZOL-4-ONES, CENTRAL BENZODIAZEPINE RECEPTOR LIGANDS

被引：33

作者：

COLOTTA, V ^{[1
]}

CECCHI, L ^{[1
]}

FILACCHIONI, G ^{[1
]}

MELANI, F ^{[1
]}

PALAZZINO, G ^{[1
]}

MARTINI, C ^{[1
]}

GIANNACCINI, G ^{[1
]}

LUCACCHINI, A ^{[1
]}

机构：

[1] UNIV PISA,IST POLICATTEDRA DISCIPLINE BIOL,I-56100 PISA,ITALY

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 01期

关键词：

D O I：

10.1021/jm00396a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1 / 3

页数：3

共 11 条

[1]

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[2]

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NADI, AI ;

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[4]

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[5] PYRAZOLO[4,5-C]QUINOLINES .3. SYNTHESIS, RECEPTOR-BINDING, AND C-13 NMR-STUDY [J].

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CECCHI, L ;

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LUCACCHINI, A .

JOURNAL OF PHARMACEUTICAL SCIENCES, 1986, 75 (12) :1175-1179

[6] PYRAZOLO[4,5-C]QUINOLINES .2. SYNTHESIS AND SPECIFIC-INHIBITION OF BENZODIAZEPINE RECEPTOR-BINDING [J].

MELANI, F ;

CECCHI, L ;

PALAZZINO, G ;

FILACCHIONI, G ;

MARTINI, C ;

PENNACCHI, E ;

LUCACCHINI, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (02) :291-295

[7]

PALAZZINO G, IN PRESS J MED CHEM

[8] CYCLO-ADDITION OF DIPHENYLNITRILIMINE TO COUMARINS - THE SYNTHESIS OF 3A,9B-DIHYDRO-4-OXO-1H-BENZOPYRANO[4,3-C]PYRAZOLE DERIVATIVES [J].

SHAWALI, AS ;

ELANADOULI, BE ;

ALBAR, HA .

TETRAHEDRON, 1985, 41 (10) :1877-1884

[9]

TYUNOSIN U, 1951, YAKUGAKU ZASSHI, V71, P857

[10]

VULFSON NS, 1961, J GEN CHEM USSR, V31, P3151

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