CARDIAC BETA-ADRENERGIC-RECEPTOR - EVALUATION OF FM 24 AS A NEW AND VERY SLOWLY DISSOCIABLE BLOCKER

被引:24
作者
LEFUR, G [1 ]
SCHMELCK, PH [1 ]
GEYNET, P [1 ]
HANOUNE, J [1 ]
UZAN, A [1 ]
机构
[1] HOP HENRI MONDOR,UNITE RECH U99,F-94010 CRETEIL,FRANCE
关键词
D O I
10.1016/0024-3205(78)90117-0
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1841 / 1850
页数:10
相关论文
共 12 条
[1]   BIOCHEMICAL EVIDENCE FOR DUAL ACTION OF LABETALOL ON ALPHA-ADRENOCEPTORS AND BETA-ADRENOCEPTORS [J].
AGGERBECK, M ;
GUELLAEN, G ;
HANOUNE, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1978, 62 (04) :543-548
[2]  
ALEXANDER W, 1975, P NATL ACAD SCI USA, V72, P1564
[3]   AFFINITY LABEL FOR BETA-ADRENERGIC-RECEPTOR IN TURKEY ERYTHROCYTES [J].
ATLAS, D ;
STEER, ML ;
LEVITZKI, A .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1976, 73 (06) :1921-1925
[4]   IRREVERSIBLE BLOCKER FOR BETA-ADRENERGIC-RECEPTOR [J].
ATLAS, D ;
LEVITZKI, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 69 (02) :397-403
[5]   POTENTIAL PROBE FOR ISOLATION OF BETA-ADRENOCEPTOR, CHLOROPRACTOLOL [J].
EREZ, M ;
WEINSTOCK, M ;
COHEN, S ;
SHTACHER, G .
NATURE, 1975, 255 (5510) :635-636
[6]  
GUELLAEN G, 1978, J BIOL CHEM, V253, P1114
[7]  
HANOUNE J, 1975, J BIOL CHEM, V250, P4569
[8]  
HANOUNE J, 1977, J BIOL CHEM, V252, P2039
[9]   CAN CHLOROPRACTOLOL ALKYLATE BETA-ADRENOCEPTORS [J].
KENAKIN, TP ;
BLACK, JW .
NATURE, 1977, 265 (5592) :365-366
[10]   PAX AND COMPETITIVE DRUG ANTAGONISM [J].
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1949, 4 (03) :277-280