SPECIFIC [H-3] SCH23390 BINDING TO DOPAMINE-D1 RECEPTORS IN CEREBRAL-CORTEX AND NEOSTRIATUM - ROLE OF DISULFIDE AND SULFHYDRYL-GROUPS

被引:24
作者
DEWAR, KM [1 ]
READER, TA [1 ]
机构
[1] UNIV MONTREAL,FAC MED,DEPT PHYSIOL,CTR RECH SCI NEUROL,CP 6128,SUCCURSALE A,MONTREAL H3C 3J7,QUEBEC,CANADA
关键词
D O I
10.1111/j.1471-4159.1989.tb09145.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:472 / 482
页数:11
相关论文
共 45 条
[1]   A COMPARISON BETWEEN DOPAMINE-STIMULATED ADENYLATE-CYCLASE AND H-3-SCH-23390 BINDING IN RAT STRIATUM [J].
ANDERSEN, PH ;
GRONVALD, FC ;
JANSEN, JA .
LIFE SCIENCES, 1985, 37 (21) :1971-1983
[2]  
ARONSTAM RS, 1978, MOL PHARMACOL, V14, P575
[3]  
BARLOW RB, 1983, BIODATA HANDLING MIC
[4]   MODULATION OF ACETYLCHOLINE-RECEPTOR STATES BY THIOL MODIFICATION [J].
BARRANTES, FJ .
BIOCHEMISTRY, 1980, 19 (13) :2957-2965
[5]   CHARACTERIZATION OF THE BINDING OF H-3-SCH 23390, A SELECTIVE D-1 RECEPTOR ANTAGONIST LIGAND, IN RAT STRIATUM [J].
BILLARD, W ;
RUPERTO, V ;
CROSBY, G ;
IORIO, LC ;
BARNETT, A .
LIFE SCIENCES, 1984, 35 (18) :1885-1893
[6]  
BOYSON SJ, 1986, J NEUROSCI, V6, P3177
[7]   EFFECTS OF HEAVY-METAL CATIONS AND OTHER SULFHYDRYL-REAGENTS ON BRAIN DOPAMINE D1 RECEPTORS - EVIDENCE FOR INVOLVEMENT OF A THIOL-GROUP IN THE CONFORMATION OF THE ACTIVE-SITE [J].
BRAESTRUP, C ;
ANDERSEN, PH .
JOURNAL OF NEUROCHEMISTRY, 1987, 48 (06) :1667-1672
[8]   STEREOSPECIFIC BINDING OF A NEW BENZAZEPINE, [H-3] SCH23390, IN CORTEX AND NEOSTRIATUM [J].
BRIERE, R ;
DIOP, L ;
GOTTBERG, E ;
GRONDIN, L ;
READER, TA .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1987, 65 (07) :1507-1511
[9]  
BZOWEJ N H, 1987, Society for Neuroscience Abstracts, V13, P1198
[10]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099