EFFECT OF THIORIDAZINE ON THE 1ST-PASS KINETICS OF [IMIPRAMINE-C-14 IN PERFUSED-RAT-LIVER - INTERACTION AT HEPATIC BINDING-SITES

被引:3
作者
BEAUBIEN, AR
PAKUTS, AP
机构
关键词
D O I
10.3109/00498258009033750
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:235 / 242
页数:8
相关论文
共 16 条
[1]  
BEAUBIEN AR, 1979, DRUG METAB DISPOS, V7, P34
[2]  
BEAUBIEN AR, 1977, PHARMACOLOGIST, V19, P128
[3]   LIVER PERFUSION TECHNIQUE USING INEXPENSIVE NON-BINDING MEDIUM FOR 1ST-PASS METABOLISM STUDIES OF DRUGS [J].
BEAUBIEN, AR ;
TRYPHONAS, L ;
PAKUTS, AP ;
MACCONAILL, M ;
COMBLEY, HA .
JOURNAL OF PHARMACOLOGICAL METHODS, 1979, 2 (03) :213-221
[4]   BINDING OF CHLORPROMAZINE AND IMIPRAMINE TO RED-CELLS, ALBUMIN, LIPOPROTEINS AND OTHER BLOOD COMPONENTS [J].
BICKEL, MH .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1975, 27 (10) :733-738
[5]   METABOLISM OF IMIPRAMINE AND ITS METABOLITES BY RAT LIVER MICROSOMES [J].
BICKEL, MH ;
BAGGIOLINI, M .
BIOCHEMICAL PHARMACOLOGY, 1966, 15 (08) :1155-+
[6]  
CRAMMER JL, 1972, PSYCHOPHARMACOLOGIA, V26, P81
[8]  
FREDRICSONOVERO K, 1977, ACTA PHARMACOL TOX, V40, P97
[9]  
FULLER RW, 1974, TOXICOL APPL PHARM, V29, P259, DOI 10.1016/0041-008X(74)90063-5
[10]  
GRAM LF, 1974, ACTA PHARMACOL TOX, V35, P223