HETEROCYCLIC GABA ANALOGS AS NEW SELECTIVE INHIBITORS OF ASTROGLIAL GABA TRANSPORT

被引:37
作者
SCHOUSBOE, A
LARSSON, OM
HERTZ, L
KROGSGAARDLARSEN, P
机构
[1] ROYAL DANISH SCH PHARM,BIOCHEM LAB,DK-2100 COPENHAGEN O,DENMARK
[2] ROYAL DANISH SCH PHARM,DEPT CHEM BC,DK-2100 COPENHAGEN O,DENMARK
[3] UNIV SASKATCHEWAN,DEPT PHARMACOL,SASKATOON S7N 0W0,SASKATCHEWAN,CANADA
关键词
D O I
10.1002/ddr.430010204
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:115 / 127
页数:13
相关论文
共 65 条
[1]  
AKKERMAN AM, 1951, RECL TRAV CHIM PAY B, V70, P899
[2]   TRANSPORT OF L-PROLINE BY RAT-BRAIN SLICES [J].
BALCAR, VJ ;
JOHNSTON, GAR ;
STEPHANSON, AL .
BRAIN RESEARCH, 1976, 102 (01) :143-151
[3]   HIGH-AFFINITY UPTAKE OF GAMMA-AMINOBUTYRIC ACID IN CULTURED GLIAL AND NEURONAL CELLS [J].
BALCAR, VJ ;
MARK, J ;
BORG, J ;
MANDEL, P .
NEUROCHEMICAL RESEARCH, 1979, 4 (03) :339-354
[4]   GABA UPTAKE IN RAT-BRAIN SLICES - INHIBITION BY GABA ANALOGS AND BY VARIOUS DRUGS [J].
BEART, PM ;
JOHNSTON, GA .
JOURNAL OF NEUROCHEMISTRY, 1973, 20 (02) :319-324
[5]   COMPETITIVE INHIBITION OF GABA UPTAKE IN RAT-BRAIN SLICES BY SOME GABA ANALOGS OF RESTRICTED CONFORMATION [J].
BEART, PM ;
JOHNSTON, GA ;
UHR, ML .
JOURNAL OF NEUROCHEMISTRY, 1972, 19 (08) :1855-&
[6]   LOCALIZING H-3-GABA IN NERVE TERMINALS OF RAT CEREBRAL CORTEX BY ELECTRON MICROSCOPIC AUTORADIOGRAPHY [J].
BLOOM, FE ;
IVERSEN, LL .
NATURE, 1971, 229 (5287) :628-&
[7]   DETERMINATION OF BRAIN-SPECIFIC ANTIGENS IN SHORT-TERM CULTIVATED RAT ASTROGLIAL CELLS AND IN RAT SYNAPTOSOMES [J].
BOCK, E ;
JORGENSEN, OS ;
DITTMANN, L ;
ENG, LF .
JOURNAL OF NEUROCHEMISTRY, 1975, 25 (06) :867-&
[8]   GLIAL FIBRILLARY ACIDIC PROTEIN IN PRIMARY ASTROGLIAL CELL-CULTURES DERIVED FROM NEWBORN RAT-BRAIN [J].
BOCK, E ;
MOLLER, M ;
NISSEN, C ;
SENSENBRENNER, M .
FEBS LETTERS, 1977, 83 (02) :207-211
[9]  
BOOHER J, 1972, Neurobiology (Copenhagen), V2, P97
[10]  
CHASE TN, 1979, A BENZON S, V12, P283