SYNTHESIS OF 1,3-DIAZEPIN-2-ONE NUCLEOSIDES AS TRANSITION-STATE INHIBITORS OF CYTIDINE DEAMINASE

被引：29

作者：

MARQUEZ, VE ^{[1
]}

LIU, PS ^{[1
]}

KELLEY, JA ^{[1
]}

DRISCOLL, JS ^{[1
]}

MCCORMACK, JJ ^{[1
]}

机构：

[1] UNIV VERMONT,COLL MED,DEPT PHARMACOL,BURLINGTON,VT 05401

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1980年 / 23卷 / 07期

关键词：

D O I：

10.1021/jm00181a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：713 / 715

页数：3

共 13 条

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[7] 1,3-DIAZEPINONES .1. SYNTHESIS OF 5-HYDROXYPERHYDRO-1,3-DIAZEPIN-2-ONE [J].

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[8] INHIBITION OF CYTIDINE DEAMINASE BY 2-OXOPYRIMIDINE RIBOSIDE AND RELATED-COMPOUNDS [J].

MCCORMACK, JJ ;

MARQUEZ, VE ;

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[9]

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[10]

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