MYOCARDIAL MUSCARINIC ACETYLCHOLINE-RECEPTOR - CHOLINE AND TRIS UNMASK HETEROGENEITY OF ANTAGONIST BINDING-SITES

被引:17
作者
SASTRE, A [1 ]
MURPHY, KMM [1 ]
RUSHER, MM [1 ]
机构
[1] JOHNS HOPKINS UNIV, SCH MED, DEPT NEUROSCI, BALTIMORE, MD 21205 USA
关键词
D O I
10.1016/0006-291X(82)90648-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:383 / 388
页数:6
相关论文
共 16 条
[1]   GUANINE-NUCLEOTIDES MODULATE MUSCARINIC RECEPTOR-BINDING IN THE HEART [J].
BERRIE, CP ;
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 87 (04) :1000-1005
[2]   CHARACTER OF THE MUSCARINIC RECEPTORS IN DIFFERENT REGIONS OF THE RAT-BRAIN [J].
BIRDSALL, NJM ;
HULME, EC ;
BURGEN, A .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1980, 207 (1166) :1-12
[3]  
BIRDSALL NJM, 1978, MOL PHARMACOL, V14, P723
[4]   EFFECTS OF IONS ON THE BINDING OF AGONISTS AND ANTAGONISTS TO MUSCARINIC RECEPTORS [J].
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC ;
WELLS, JW .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 67 (03) :371-377
[5]  
Dale HH, 1914, J PHARMACOL EXP THER, V6, P147
[6]  
FIELDS JZ, 1978, J BIOL CHEM, V253, P3251
[7]  
HAUBRICH DR, 1979, BIOCHEM PHARMACOL, V28, P3673, DOI 10.1016/0006-2952(79)90417-9
[8]  
HULME EC, 1978, MOL PHARMACOL, V14, P737
[9]   MUSCARINIC ACETYLCHOLINE RECEPTORS INTERACTIONS - COMPETITION BINDING STUDIES WITH AGONISTS AND ANTAGONISTS [J].
KLOOG, Y ;
SOKOLOVSKY, M .
BRAIN RESEARCH, 1977, 134 (01) :167-172
[10]   CHOLINE EXCITES CORTICAL-NEURONS [J].
KRNJEVIC, K ;
REINHARDT, W .
SCIENCE, 1979, 206 (4424) :1321-1323