EFFICIENT SYNTHESIS OF 3-SUBSTITUTED INDOLES BY PALLADIUM-CATALYZED COUPLING REACTION OF 3-TRIBUTYLSTANNYLINDOLES WITH ORGANIC TRIFLATES AND HALIDES

被引：49

作者：

CIATTINI, PG

MORERA, E

ORTAR, G

机构：

[1] UNIV ROMA LA SAPIENZA,CNR,DIPARTIMENTO STUDI FARMACEUT,I-00185 ROME,ITALY

[2] UNIV ROMA LA SAPIENZA,CNR,CTR STUDIO CHIM FARMACO,I-00185 ROME,ITALY

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 15期

关键词：

D O I：

10.1016/0040-4039(94)85231-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The palladium-catalyzed reaction of 1-tosyl-3-tributylstannylindoles 2 with a variety of vinyl, aryl, and heteroaryl triflates and halides (1) provides a general and efficient method for the synthesis of 3-substituted indoles 3.

引用

页码：2405 / 2408

页数：4

共 24 条

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