IRREVERSIBLE SELECTIVE BLOCKADE OF KAPPA-OPIOID RECEPTORS IN THE GUINEA-PIG ILEUM

被引：13

作者：

SHEEHAN, MJ

HAYES, AG

TYERS, MB

机构：

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY | 1986年 / 129卷 / 1-2期

关键词：

D O I：

10.1016/0014-2999(86)90331-6

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：19 / 24

页数：6

共 14 条

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[3]

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[6]

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[8] 6-BETA [N,N-BIS(2-CHLOROETHYL)AMINO]-17-(CYCLOPROPYLMETHYL)-4,5-ALPHA-EPOXY-3,14-DIHYDROXYMORPHINAN (CHLORANALTREXAMINE) - POTENT OPIOID RECEPTOR ALKYLATING AGENT WITH ULTRALONG NARCOTIC-ANTAGONIST ACTIVITY [J].

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[10] NOVEL OPIOID RECEPTOR-SITE DIRECTED ALKYLATING AGENT WITH IRREVERSIBLE NARCOTIC ANTAGONISTIC AND REVERSIBLE AGONISTIC ACTIVITIES [J].

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