THE UNIT IMPULSE-RESPONSE PROCEDURE FOR THE PHARMACOKINETIC EVALUATION OF DRUG ENTRY INTO THE CENTRAL NERVOUS-SYSTEM

被引:29
作者
VANBREE, JBMM
BALJET, AV
VANGEYT, A
DEBOER, AG
DANHOF, M
BREIMER, DD
机构
来源
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS | 1989年 / 17卷 / 04期
关键词
D O I
10.1007/BF01061457
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:441 / 462
页数:22
相关论文
共 29 条
[1]   PERMEABILITY OF THE BLOOD-BRAIN-BARRIER TO NEUROPEPTIDES - THE CASE FOR PENETRATION [J].
BANKS, WA ;
KASTIN, AJ .
PSYCHONEUROENDOCRINOLOGY, 1985, 10 (04) :385-399
[2]  
BERING EA, 1974, FED PROC, V33, P2061
[3]   RAPID AND SIMPLE CANNULATION TECHNIQUE FOR REPEATED SAMPLING OF CEREBROSPINAL-FLUID IN FREELY MOVING RATS [J].
BOUMAN, HJ ;
VANWIMERSMAGREIDANUS, TB .
BRAIN RESEARCH BULLETIN, 1979, 4 (04) :575-577
[4]  
BRODIE BB, 1960, J PHARMACOL EXP THER, V130, P519
[5]   DISTRIBUTED MODEL FOR DRUG DELIVERY TO CSF AND BRAIN-TISSUE [J].
COLLINS, JM ;
DEDRICK, RL .
AMERICAN JOURNAL OF PHYSIOLOGY, 1983, 245 (03) :R303-R310
[6]   PERMEABILITY OF CAPILLARIES IN VARIOUS ORGANS AS DETERMINED BY USE OF INDICATOR DIFFUSION METHOD [J].
CRONE, C .
ACTA PHYSIOLOGICA SCANDINAVICA, 1963, 58 (04) :292-&
[7]  
DANHOF M, 1984, J PHARMACOL EXP THER, V229, P44
[8]  
DAVSON H, 1976, J PHYSIOL-LONDON, V255, P1
[9]   PHARMACOKINETIC MODELING OF THE ANTICONVULSANT RESPONSE OF OXAZEPAM IN RATS USING THE PENTYLENETETRAZOL THRESHOLD CONCENTRATION AS PHARMACODYNAMIC MEASURE [J].
DINGEMANSE, J ;
SOLLIE, FAE ;
BREIMER, DD ;
DANHOF, M .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1988, 16 (02) :203-228
[10]   METHODS FOR QUANTIFYING THE TRANSPORT OF DRUGS ACROSS BRAIN BARRIER SYSTEMS [J].
FENSTERMACHER, JD ;
BLASBERG, RG ;
PLATLAK, CS .
PHARMACOLOGY & THERAPEUTICS, 1981, 14 (02) :217-248