BASE-MODIFIED PYRIMIDINE NUCLEOSIDES - EFFICIENT ENTRY TO 6-DERIVATIZED URIDINES BY SN-PD TRANSMETALATION-COUPLING PROCESS

被引：40

作者：

PALMISANO, G ^{[1
]}

SANTAGOSTINO, M ^{[1
]}

机构：

[1] CNR,CTR STUDIO SOSTANZE ORGAN NAT,I-20133 MILAN,ITALY

来源：

TETRAHEDRON | 1993年 / 49卷 / 12期

关键词：

D O I：

10.1016/S0040-4020(01)86332-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The palladium-catalyzed reaction of 6-tributylstannyluridine derivative 5 with a variety of aryl, vinyl, alkynyl, and allyl halides provides an efficient method for the synthesis of the corresponding cross-coupled products. In all cases, an enhancement on the rate and isolated yields was attained by using Cul as co-catalyst.

引用

页码：2533 / 2542

页数：10

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