SYNTHESIS OF A MORPHINE-6-GLUCURONIDE HAPTEN, N-(4-AMINOBUTYL)NORMORPHINE-6-GLUCURONID AND RELATED HAPTENS

被引：25

作者：

BROWN, RT ^{[1
]}

CARTER, NE ^{[1
]}

LUMBARD, KW ^{[1
]}

SCHEINMANN, F ^{[1
]}

机构：

[1] SALFORD ULTRAFINE CHEM & RES LTD,MANCHESTER M15 6SY,LANCS,ENGLAND

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 47期

关键词：

D O I：

10.1016/0040-4039(95)01786-H

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

For use as a hapten in the radioimmunoassay of morphine-6-glucuronide 2 (M6G), N-(4-aminobutyl)normorphine-6-glucuronide 12 has been prepared, together with related haptens, using the imidate coupling method developed for synthesis of M6G; a rebuttal of recent critical comments on our synthesis of M6G is included.

引用

页码：8661 / 8664

页数：4

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