MIXED TYPE INHIBITION OF [D-ALA2,D-LEU5]ENKEPHALIN BINDING TO MU-OPIATE BINDING-SITES BY MU-, BUT NOT BY KAPPA-OPIATE LIGANDS

被引:3
作者
PFEIFFER, A [1 ]
HERZ, A [1 ]
机构
[1] MAX PLANCK INST PSYCHIAT,DEPT NEUROPHARMACOL,D-8000 MUNICH 40,FED REP GER
关键词
D O I
10.1016/0014-2999(82)90145-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:359 / 361
页数:3
相关论文
共 7 条
[1]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[2]   DIFFERENTIATION OF DELTA AND MU OPIATE RECEPTOR LOCALIZATIONS BY LIGHT MICROSCOPIC AUTORADIOGRAPHY [J].
GOODMAN, RR ;
SNYDER, SH ;
KUHAR, MJ ;
YOUNG, WS .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (10) :6239-6243
[3]   CHARACTERIZATION OF THE KAPPA-SUBTYPE OF THE OPIATE RECEPTOR IN THE GUINEA-PIG BRAIN [J].
KOSTERLITZ, HW ;
PATERSON, SJ ;
ROBSON, LE .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 73 (04) :939-949
[4]   ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].
LORD, JAH ;
WATERFIELD, AA ;
HUGHES, J ;
KOSTERLITZ, HW .
NATURE, 1977, 267 (5611) :495-499
[5]  
MARTIN WR, 1976, J PHARMACOL EXP THER, V197, P517
[6]   DEMONSTRATION AND DISTRIBUTION OF AN OPIATE BINDING-SITE IN RAT-BRAIN WITH HIGH-AFFINITY FOR ETHYLKETOCYCLAZOCINE AND SKF 10,047 [J].
PFEIFFER, A ;
HERZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 101 (01) :38-44
[7]  
PFEIFFER A, 1981, Naunyn-Schmiedeberg's Archives of Pharmacology, V316, pR61