PEPTOIDS - A NEW APPROACH TO THE DEVELOPMENT OF PHARMACEUTICALS

被引：97

作者：

KESSLER, H

机构：

[1] Organisch-Chemisches Institut, Technischen Universität München, Garching, D-W-8046

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1993年 / 32卷 / 04期

关键词：

D O I：

10.1002/anie.199305431

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

N‐substituted oligoglycines, “peptoids”, can be prepared in good yields and high purity without protected monomer building blocks and without deprotection according to Equation (a). This class of compounds should be of great utility in screening for new pharmaceutical lead structures. (Figure Presented.) Copyright © 1993 by VCH Verlagsgesellschaft mbH, Germany

引用

页码：543 / 544

页数：2

共 12 条

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[10] PEPTOIDS - A MODULAR APPROACH TO DRUG DISCOVERY
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JEWELL, DA
BANVILLE, S
NG, S
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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (20) : 9367 - 9371

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