SYNTHESIS OF 7,12-DIHYDRO-INDOLO[3,2-D][1]BENZAZEPIN-6-(5H)-ONES AND 6,11-DIHYDRO-THIENO[3',2'/2,3]AZEPINO[4,5-B]INDOL-5(4H)-ONE

被引：34

作者：

KUNICK, C

机构：

[1] Pharmazeutisches Institut, Universität Bonn, Bonn, D-5300

来源：

ARCHIV DER PHARMAZIE | 1992年 / 325卷 / 05期

关键词：

D O I：

10.1002/ardp.19923250509

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The title compounds 4 and 6 were prepared by Fischer indole synthesis. 4a is substituted in 10-position by reaction with bromine in glacial acetic acid. A fast ring inversion is observed for the azepine ring in 4 and 6.

引用

页码：297 / 299

页数：3

共 6 条

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[6]

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