ARYL RADICAL CYCLIZATION APPROACH TO HIGHLY SUBSTITUTED OXINDOLES RELATED TO MITOMYCINS

被引：15

作者：

JONES, K

STOREY, JMD

机构：

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 48期

关键词：

ARYL RADICAL CYCLIZATION; OXINDOLES; MITOMYCINS;

D O I：

10.1016/S0040-4039(00)61569-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Radical cyclisation of the hexa-substituted aromatic compounds 8 and 17 leads to highly substituted oxindoles 9 and 18 respectively in excellent yields. Oxindole 18 carries the correct substitution pattern for ring-A of mitomycin A.

引用

页码：7797 / 7798

页数：2

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