SYNTHESIS OF BOXAZOMYCIN B AND RELATED ANALOGS

被引:15
作者
SUTO, MJ [1 ]
TURNER, WR [1 ]
机构
[1] WARNER LAMBERT PARKE DAVIS,PARKE DAVIS PHARMACEUT RES DIV,DEPT CHEM,ANN ARBOR,MI 48105
关键词
D O I
10.1016/0040-4039(95)01533-N
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The total synthesis of the novel antibacterial agent Boxazomycin B is reported. The synthesis proceeds through a highly functionalized benzene ring in which the key functionalities are introduced early in the synthesis and serve as protecting groups for additional transformations.
引用
收藏
页码:7213 / 7216
页数:4
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