DISPOSITION OF A NEW, NONSTEROID, ANTIANDROGEN, ALPHA,ALPHA,ALPHA-TRIFLUORO-2-METHYL-4'-NITRO-M-PROPIONOTOLUIDIDE (FLUTAMIDE), IN MEN FOLLOWING A SINGLE ORAL 200 MG DOSE

被引:118
作者
KATCHEN, B [1 ]
BUXBAUM, S [1 ]
机构
[1] SCHERING CORP, DEPT BIOCHEM, BIOL RES DIV, BLOOMFIELD, NJ 07703 USA
关键词
D O I
10.1210/jcem-41-2-373
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:373 / 379
页数:7
相关论文
共 7 条
[1]   ACTION OF A NONSTEROIDAL ANTIANDROGEN, FLUTAMIDE, ON RECEPTOR-BINDING AND NUCLEAR RETENTION OF 5-ALPHA DIHYDROTESTOSTERONE IN RAT VENTRAL PROSTATE [J].
LIAO, S ;
HOWELL, DK ;
CHANG, TM .
ENDOCRINOLOGY, 1974, 94 (04) :1205-1209
[2]   INVESTIGATION INTO ANTI-ANDROGENIC PROPERTIES OF NONSTEROIDAL COMPOUND, SCH 13521 (4'-NITRO-3'-TRIFLUOROMETHYLISOBUTYRYLANILIDE) [J].
MAINWARING, WI ;
MANGAN, FR ;
FEHERTY, PA ;
FREIFELD, M .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1974, 1 (02) :113-128
[3]   BIOLOGICAL PROFILE OF A NONSTEROIDAL ANTIANDROGEN, SCH 13521 4'-NITRO-3'-TRIFLUOROMETHYLISOBUTYRANILIDE [J].
NERI, R ;
VANCLEAV.S ;
FLORANCE, K ;
KOZIOL, P .
ENDOCRINOLOGY, 1972, 91 (02) :427-&
[4]  
NERI RO, 1972, INVEST UROL, V10, P123
[5]   MECHANISM OF ANTIANDROGENIC ACTION OF GLUTAMIDE (ALPHA-ALPHA-ALPHA-TRIFLUORO-2-METHYL-4'-NITRO-M-PROPIONOTOLUIDIDE) IN RAT [J].
PEETS, EA ;
HENSON, MF ;
NERI, R .
ENDOCRINOLOGY, 1974, 94 (02) :532-540
[6]   PHYSIOLOGY AND TOXICOLOGY OF TRITIUM IN MAN [J].
PINSON, EA ;
LANGHAM, WH .
JOURNAL OF APPLIED PHYSIOLOGY, 1957, 10 (01) :108-126
[7]   SCH-13521 IN TREATMENT OF ADVANCED CARCINOMA OF PROSTATE [J].
STOLIAR, B ;
ALBERT, DJ .
JOURNAL OF UROLOGY, 1974, 111 (06) :803-807