SLOW-BINDING AND FAST-BINDING INHIBITORS OF THERMOLYSIN DISPLAY DIFFERENT MODES OF BINDING - CRYSTALLOGRAPHIC ANALYSIS OF EXTENDED PHOSPHONAMIDATE TRANSITION-STATE ANALOGS

被引：216

作者：

HOLDEN, HM

TRONRUD, DE

MONZINGO, AF

WEAVER, LH

MATTHEWS, BW

机构：

[1] UNIV OREGON,INST MOLEC BIOL,EUGENE,OR 97403

[2] UNIV OREGON,DEPT PHYS,EUGENE,OR 97403

来源：

BIOCHEMISTRY | 1987年 / 26卷 / 26期

关键词：

D O I：

10.1021/bi00400a008

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：8542 / 8553

页数：12

共 49 条

[1]

ANTONOV VK, 1981, EUR J BIOCHEM, V117, P195

[2] SIMILARITIES IN ACTIVE-CENTER GEOMETRIES OF ZINC-CONTAINING ENZYMES, PROTEASES AND DEHYDROGENASES [J].

ARGOS, P ;

GARAVITO, RM ;

EVENTOFF, W ;

ROSSMANN, MG ;

BRANDEN, CI .

JOURNAL OF MOLECULAR BIOLOGY, 1978, 126 (02) :141-158

[3] POSSIBLE ROLE FOR WATER DISSOCIATION IN THE SLOW BINDING OF PHOSPHORUS-CONTAINING TRANSITION-STATE-ANALOGUE INHIBITORS OF THERMOLYSIN [J].

BARTLETT, PA ;

MARLOWE, CK .

BIOCHEMISTRY, 1987, 26 (26) :8553-8561

[4] PHOSPHONAMIDATES AS TRANSITION-STATE ANALOG INHIBITORS OF THERMOLYSIN [J].

BARTLETT, PA ;

MARLOWE, CK .

BIOCHEMISTRY, 1983, 22 (20) :4618-4624

[5]

BOLOGNESI MC, 1979, J BIOL CHEM, V254, P634

[6]

Bowen H.J.M., 1958, TABLES INTERATOMIC D

[7] X-RAY CRYSTALLOGRAPHIC INVESTIGATION OF SUBSTRATE BINDING TO CARBOXYPEPTIDASE-A AT SUBZERO TEMPERATURE [J].

CHRISTIANSON, DW ;

LIPSCOMB, WN .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (20) :7568-7572

[8] ADENOSINE-DEAMINASE AND ADENYLATE DEAMINASE - COMPARATIVE KINETIC-STUDIES WITH TRANSITION-STATE AND GROUND-STATE ANALOG INHIBITORS [J].

FRIEDEN, C ;

KURZ, LC ;

GILBERT, HR .

BIOCHEMISTRY, 1980, 19 (23) :5303-5309

[9] INHIBITION OF ANGIOTENSIN CONVERTING ENZYME BY PHOSPHORAMIDATES AND POLYPHOSPHATES [J].

GALARDY, RE .

BIOCHEMISTRY, 1982, 21 (23) :5777-5781

[10] INHIBITION OF ANGIOTENSIN CONVERTING ENZYME BY PHOSPHONIC AMIDES AND PHOSPHONIC-ACIDS [J].

GALARDY, RE ;

KONTOYIANNIDOUOSTREM, V ;

KORTYLEWICZ, ZP .

BIOCHEMISTRY, 1983, 22 (08) :1990-1995

← 1 2 3 4 5 →