PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .19. SYNTHESIS OF (+)-4-[(ALPHA-R)-ALPHA-((2S,5R)-4-ALLYL-2,5-DIMETHYL-1-PIPERAZINYL)-3-METHOXYBENZYL]-N,N-DIETHYLBENZAMIDE (SNC-80) - A HIGHLY SELECTIVE, NONPEPTIDE DELTA-OPIOID RECEPTOR AGONIST

被引：198

作者：

CALDERON, SN

ROTHMAN, RB

PORRECA, F

FLIPPENANDERSON, JL

MCNUTT, RW

XU, H

SMITH, LE

BILSKY, EJ

DAVIS, P

RICE, KC

机构：

[1] NIDDKD,MED CHEM LAB,BETHESDA,MD 20892

[2] NIDA,ADDICT RES CTR,CLIN PSYCHOPHARMACOL SECT,BALTIMORE,MD 21224

[3] USN,RES LAB,STRUCT MATTER LAB,CODE 6030,WASHINGTON,DC 20375

[4] UNIV ARIZONA,ARIZONA HLTH SCI CTR,DEPT PHARMACOL,TUCSON,AZ 85724

[5] BURROUGHS WELLCOME CO,DIV ORGAN CHEM,RES TRIANGLE PK,NC 27709

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 14期

关键词：

D O I：

10.1021/jm00040a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：2125 / 2128

页数：4

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