PREPARATION OF N-ALKYL PYRROLIDINONES VIA PHOTOCYCLIZATION OF GAMMA-KETO-ALPHA,BETA-UNSATURATED AMIDES

被引：19

作者：

DITTAMI, JP ^{[1
]}

XU, F ^{[1
]}

QI, H ^{[1
]}

MARTIN, MW ^{[1
]}

BORDNER, J ^{[1
]}

DECOSTA, DL ^{[1
]}

KIPLINGER, J ^{[1
]}

REICHE, P ^{[1
]}

WARE, R ^{[1
]}

机构：

[1] PFIZER INC,CENT RES,GROTON,CT 06340

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 24期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/0040-4039(95)00779-C

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Photolysis of gamma-keto-alpha,beta-unsaturated amides provides N-alkyl pyrrolidinones in high yield (77-100%). The procedure is applicable to a variety of amides derived from the corresponding gamma-keto acid.

引用

页码：4197 / 4200

页数：4

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