SYNTHESES OF HOMOSERINE PHOSPHATE ANALOGS AS POTENTIAL INHIBITORS OF BACTERIAL THREONINE SYNTHASE

被引：16

作者：

HARDE, C

NEFF, KH

NORDHOFF, E

GERBLING, KP

LABER, B

POHLENZ, HD

机构：

[1] Schering AG, Agrochemical Research

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1994年 / 4卷 / 02期

关键词：

D O I：

10.1016/S0960-894X(01)80128-1

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The syntheses of five homoserine phosphate analogs (1-4, Z-5) are described. A brief summary of their potential to inhibit threonine synthase from Escherichia coli is given.

引用

页码：273 / 278

页数：6

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