PHARMACOLOGY OF SOME METABOLITES OF TRIAZOLAM, ALPRAZOLAM, AND DIAZEPAM PREPARED BY A SIMPLE, ONE-STEP OXIDATION OF BENZODIAZEPINES

被引：49

作者：

GALL, M

KAMDAR, BV

COLLINS, RJ

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1978年 / 21卷 / 12期

关键词：

D O I：

10.1021/jm00210a022

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1290 / 1294

页数：5

共 30 条

[1] QUINAZOLINES + 1,4-BENZODIAZEPINES .16. SYNTHESIS + TRANSFORMATIONS OF 5-PHENYL-1,4-BENZODIAZEPINE-2-THIONES [J].

ARCHER, GA ;

STERNBACH, LH .

JOURNAL OF ORGANIC CHEMISTRY, 1964, 29 (01) :231-&

[2]

BARLEY EJ, 1962, J CHEM SOC, P1578

[3] A GENERAL METHOD FOR PREPARING 2-ACETAMIDOACETANILIDES HAVING A 2ND FUNCTIONAL GROUP IN 2 POSITION AND AFFORDING AN ACCESS TO 3-ACETAMIDO-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONES [J].

BELL, SC ;

MCCAULLY, RJ ;

CHILDRES.SJ .

JOURNAL OF ORGANIC CHEMISTRY, 1968, 33 (01) :216-&

[4] 3-SUBSTITUTED 1,4-BENZODIAZEPIN-2-ONES [J].

BELL, SC ;

MCCAULLY, RJ ;

GOCHMAN, C ;

CHILDRESS, SJ ;

GLUCKMAN, MI .

JOURNAL OF MEDICINAL CHEMISTRY, 1968, 11 (03) :457-+

[5] A REARRANGEMENT OF 5-ARYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPINE-2-14-OXIDES [J].

BELL, SC ;

CHILDRESS, SJ .

JOURNAL OF ORGANIC CHEMISTRY, 1962, 27 (05) :1691-&

[6] REARRANGEMENT OF 2-AMINO-5-PHENYL-3H-1,4-BENZODIAZEPINE 4-OXIDES WITH ACETIC ANHYDRIDE [J].

BELL, SC ;

GOCHMAN, C ;

CHILDRESS, SJ .

JOURNAL OF ORGANIC CHEMISTRY, 1963, 28 (11) :3010-&

[7]

BUCHI G, 1968, J AM CHEM SOC, V90, P2448

[8]

Buchi G, 1970, J Am Chem Soc, V92, P999

[9] STEREOCHEMISTRY OF ENZYMIC 3-HYDROXYLATION OF 1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONES [J].

CORBELLA, A ;

GARIBOLDI, P ;

JOMMI, G ;

FORGIONE, A ;

MARCUCCI, F ;

MARTELLI, P ;

MUSSINI, E ;

MAURI, F .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1973, (19) :721-722

[10]

EBERTS FS, 1973, FED PROC, V32, P747

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