SYNTHESIS AND REACTIONS OF LITHIATED MONOCYCLIC AZOLES CONTAINING 2 OR MORE HETERO-ATOMS .5. ISOTHIAZOLES AND THIAZOLES

被引：22

作者：

IDDON, B

机构：

[1] The Ramage Laboratories, Department of Chemistry and Applied Chemistry, University of Salford, Salford

来源：

HETEROCYCLES | 1995年 / 41卷 / 03期

关键词：

D O I：

10.3987/REV-94-466

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The metallation and halogen --> metal exchange reactions of isothiazoles (1,2-thiazoles) and thiazoles (1,3-thiazoles) and the reactions of the resulting organometallic derivatives, particularly lithiated derivatives, are reviewed comprehensively.

引用

页码：533 / 593

页数：61

共 137 条

[1] ALKYLATION OF 3,5-DIMETHYLISOTHIAZOLE - A REGIOSELECTIVE SYNTHESIS OF 5-ALKYL-3-METHYLISOTHIAZOLES [J].

ALBEROLA, A ;

ANDRES, C ;

CASADO, JL ;

GONZALEZ, A ;

PEDROSA, R .

SYNTHETIC COMMUNICATIONS, 1990, 20 (04) :617-624

[2]

ALBEROLA A, 1987, GAZZ CHIM ITAL, V117, P461

[3]

ALTMAN LJ, 1971, TETRAHEDRON LETT, P4709

[4]

APSIMON J, 1977, HETEROCYCLES, V6, P731

[5] THIAZOLE AND IMIDAZOLE METABOLITES FROM THE ASCIDIAN APLYDIUM-PLICIFERUM [J].

ARABSHAHI, L ;

SCHMITZ, FJ .

TETRAHEDRON LETTERS, 1988, 29 (10) :1099-1102

[6]

ASHTON MJ, 1984, J MED CHEM, V27, P1245, DOI 10.1021/jm00376a002

[7] AZOLES .9. SYNTHESIS OF DERIVATIVES OF THIENO[2,3-D]THIAZOLE, 4H-PYRROLO-[2,3-D]THIAZOLE, 2H-PYRAZOLO[3,4-D]THIAZOLE AND ISOXAZOLO[3,4-D]THIAZOLE FROM THIAZOLIDINE-2,4-DIONE [J].

ATHMANI, S ;

FARHAT, MF ;

IDDON, B .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1992, (08) :973-977

[8] AZOLES .8. METALATION AND BROMINE-] LITHIUM EXCHANGE-REACTIONS OF POLYHALOGENOTHIAZOLES [J].

ATHMANI, S ;

BRUCE, A ;

IDDON, B .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1992, (02) :215-219

[9]

BAKER R, 1988, Patent No. 3071412

[10] NEW METHODS FOR THE INTRODUCTION OF SUBSTITUENTS INTO THIAZOLES [J].

BEGTRUP, M ;

HANSEN, LBL .

ACTA CHEMICA SCANDINAVICA, 1992, 46 (04) :372-383

← 1 2 3 4 5 6 7 8 9 10 →