REGULATION OF THROMBOXANE RECEPTOR ACTIVATION IN HUMAN-PLATELETS

被引:100
作者
MURRAY, R [1 ]
FITZGERALD, GA [1 ]
机构
[1] VANDERBILT UNIV,DIV CLIN PHARMACOL,NASHVILLE,TN 37232
关键词
D O I
10.1073/pnas.86.1.124
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:124 / 128
页数:5
相关论文
共 29 条
[1]   INTERACTION OF STABLE PROSTAGLANDIN ENDOPEROXIDE ANALOGS U46619 AND U44069 WITH HUMAN-PLATELET MEMBRANES - COUPLING OF RECEPTORS WITH HIGH-AFFINITY GTPASE AND ADENYLATE-CYCLASE [J].
AVDONIN, PV ;
SVITINAULITINA, IV ;
LEYTIN, VL ;
TKACHUK, VA .
THROMBOSIS RESEARCH, 1985, 40 (01) :101-112
[2]   INOSITOL 1,4,5-TRIPHOSPHATE-INDUCED GRANULE SECRETION IN PLATELETS - EVIDENCE THAT THE ACTIVATION OF PHOSPHOLIPASE-C MEDIATED BY PLATELET THROMBOXANE RECEPTORS INVOLVES A GUANINE-NUCLEOTIDE BINDING PROTEIN-DEPENDENT MECHANISM DISTINCT FROM THAT OF THROMBIN [J].
BRASS, LF ;
SHALLER, CC ;
BELMONTE, EJ .
JOURNAL OF CLINICAL INVESTIGATION, 1987, 79 (04) :1269-1275
[3]   PLATELET DESENSITIZATION INDUCED BY ARACHIDONIC-ACID IS NOT DUE TO CYCLO-OXYGENASE INACTIVATION AND INVOLVES THE ENDOPEROXIDE RECEPTOR [J].
CARMO, LG ;
HATMI, M ;
ROTILIO, D ;
VARGAFTIG, BB .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 85 (04) :849-859
[4]   ACTIVATION OF TURKEY ERYTHROCYTE ADENYLATE-CYCLASE AND BLOCKING OF CATECHOLAMINE-STIMULATED GTPASE BY GUANOSINE 5'-(GAMMA-THIO) TRIPHOSPHATE [J].
CASSEL, D ;
SELINGER, Z .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 77 (03) :868-873
[5]   COMPARISON OF THE ACTIONS OF U-46619, A PROSTAGLANDIN H2-ANALOGUE, WITH THOSE OF PROSTAGLANDIN-H2 AND THROMBOXANE-A2 ON SOME ISOLATED SMOOTH-MUSCLE PREPARATIONS [J].
COLEMAN, RA ;
HUMPHREY, PPA ;
KENNEDY, I ;
LEVY, GP ;
LUMLEY, P .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 73 (03) :773-778
[6]   ENDOGENOUS BIOSYNTHESIS OF PROSTACYCLIN AND THROMBOXANE AND PLATELET-FUNCTION DURING CHRONIC ADMINISTRATION OF ASPIRIN IN MAN [J].
FITZGERALD, GA ;
OATES, JA ;
HAWIGER, J ;
MAAS, RL ;
ROBERTS, LJ ;
LAWSON, JA ;
BRASH, AR .
JOURNAL OF CLINICAL INVESTIGATION, 1983, 71 (03) :676-688
[7]  
GRYNKIEWICZ G, 1985, J BIOL CHEM, V260, P3440
[8]   A NOVEL-APPROACH FOR THE STUDY OF THROMBOXANE-A2 AND PROSTAGLANDIN-H2 RECEPTORS USING AN I-125-LABELED LIGAND [J].
HALUSHKA, PV ;
MACDERMOT, J ;
KNAPP, DR ;
ELLER, T ;
SAUSSY, DL ;
MAIS, D ;
BLAIR, IA ;
DOLLERY, CT .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (08) :1165-1170
[9]   THROMBOXANES - NEW GROUP OF BIOLOGICALLY-ACTIVE COMPOUNDS DERIVED FROM PROSTAGLANDIN ENDOPEROXIDES [J].
HAMBERG, M ;
SVENSSON, J ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1975, 72 (08) :2994-2998
[10]  
HARDEN TK, 1983, PHARMACOL REV, V35, P5