EVIDENCE THAT THE M2 MEMBRANE-SPANNING REGION LINES THE ION CHANNEL PORE OF THE NICOTINIC RECEPTOR

被引:330
作者
LEONARD, RJ
LABARCA, CG
CHARNET, P
DAVIDSON, N
LESTER, HA
机构
关键词
D O I
10.1126/science.2462281
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1578 / 1581
页数:4
相关论文
共 40 条
[1]   KINETICS OF AGONIST CONDUCTANCE CHANGES DURING HYPERPOLARIZATION AT FROG ENDPLATES [J].
ADAMS, PR .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (02) :308-310
[2]   VOLTAGE JUMP ANALYSIS OF PROCAINE ACTION AT FROG ENDPLATE [J].
ADAMS, PR .
JOURNAL OF PHYSIOLOGY-LONDON, 1977, 268 (02) :291-318
[3]  
ADAMS PR, 1975, PFLUG ARCH EUR J PHY, V360, P155, DOI 10.1007/BF00580538
[4]  
ADLER M, 1978, MOL PHARMACOL, V14, P514
[5]  
ARACAVA Y, 1984, MOL PHARM, V26, P293
[6]   QUANTITATIVE DESCRIPTION OF ENDPLATE CURRENTS IN PRESENCE OF 2 LIDOCAINE DERIVATIVES [J].
BEAM, KG .
JOURNAL OF PHYSIOLOGY-LONDON, 1976, 258 (02) :301-322
[7]   EFFECTS OF CHLORPROMAZINE AND PHENCYCLIDINE ON MOUSE C2 ACETYLCHOLINE-RECEPTOR KINETICS [J].
CHANGEUX, JP ;
PINSET, C ;
RIBERA, AB .
JOURNAL OF PHYSIOLOGY-LONDON, 1986, 378 :497-513
[8]  
DAHLBOM R, 1965, ACTA PHARM SUEC, V2, P213
[9]   STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - SERINE-262 OF THE DELTA-SUBUNIT IS LABELED BY [H-3] CHLORPROMAZINE [J].
GIRAUDAT, J ;
DENNIS, M ;
HEIDMANN, T ;
CHANG, JY ;
CHANGEUX, JP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (08) :2719-2723
[10]   STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - (H-3) CHLORPROMAZINE LABELS HOMOLOGOUS RESIDUES IN THE BETA-CHAIN AND DELTA-CHAIN [J].
GIRAUDAT, J ;
DENNIS, M ;
HEIDMANN, T ;
HAUMONT, PY ;
LEDERER, F ;
CHANGEUX, JP .
BIOCHEMISTRY, 1987, 26 (09) :2410-2418