DISSOCIATED EFFECTS OF INHIBITORS OF ENKEPHALIN-METABOLIZING PEPTIDASES OR NALOXONE ON VARIOUS NOCICEPTIVE RESPONSES

被引:60
作者
COSTENTIN, J [1 ]
VLAICULESCU, A [1 ]
CHAILLET, P [1 ]
BENNATAN [1 ]
AVEAUX, D [1 ]
SCHWARTZ, JC [1 ]
机构
[1] INSERM, CTR PAUL BROCA, UNITE NEUROBIOL 109, F-75014 PARIS, FRANCE
关键词
D O I
10.1016/0014-2999(86)90684-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:37 / 44
页数:8
相关论文
共 43 条
  • [1] INHIBITION OF ENKEPHALIN-DEGRADING AMINOPEPTIDASE ACTIVITY BY CERTAIN PEPTIDES
    BARCLAY, RK
    PHILLIPPS, MA
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 96 (04) : 1732 - 1738
  • [2] BENBASSAT J, 1959, ARCH INT PHARMACOD T, V122, P434
  • [3] COMPARISON OF ANALGESIC PROPERTIES OF LIPOTROPIN C-FRAGMENT AND STABILIZED ENKEPHALINS IN RAT
    BRADBURY, AF
    SMYTH, DG
    SNELL, CR
    DEAKIN, JFW
    WENDLANDT, S
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 74 (02) : 748 - 754
  • [4] EFFECT OF INHIBITION OF NEUROPEPTIDASES ON THE PAIN THRESHOLD OF MICE AND RATS
    CARENZI, A
    FRIGENI, V
    REGGIANI, A
    DELLABELLA, D
    [J]. NEUROPHARMACOLOGY, 1983, 22 (11) : 1315 - 1319
  • [5] INHIBITION OF ENKEPHALIN METABOLISM BY, AND ANTI-NOCICEPTIVE ACTIVITY OF, BESTATIN, AN AMINOPEPTIDASE INHIBITOR
    CHAILLET, P
    MARCAISCOLLADO, H
    COSTENTIN, J
    YI, CC
    DELABAUME, S
    SCHWARTZ, JC
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 86 (3-4) : 329 - 336
  • [6] CHIPKIN RE, 1982, REGUL PEPTIDES, P235
  • [7] D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
  • [8] PARTICIPATION OF BOTH ENKEPHALINASE AND AMINOPEPTIDASE ACTIVITIES IN THE METABOLISM OF ENDOGENOUS ENKEPHALINS
    DELABAUME, S
    YI, CC
    SCHWARTZ, JC
    CHAILLET, P
    MARCAISCOLLADO, H
    COSTENTIN, J
    [J]. NEUROSCIENCE, 1983, 8 (01) : 143 - 151
  • [9] PAIN MODULATION BY ADRENERGIC AGENTS AND MORPHINE AS MEASURED BY 3 PAIN TESTS
    DENNIS, SG
    MELZACK, R
    GUTMAN, S
    BOUCHER, F
    [J]. LIFE SCIENCES, 1980, 26 (15) : 1247 - 1259
  • [10] PAIN MODULATION BY 5-HYDROXYTRYPTAMINERGIC AGENTS AND MORPHINE AS MEASURED BY 3 PAIN TESTS
    DENNIS, SG
    MELZACK, R
    [J]. EXPERIMENTAL NEUROLOGY, 1980, 69 (02) : 260 - 270