ON THE ADENOSINE RECEPTOR INVOLVED IN THE EXCITATORY ACTION OF ADENOSINE ON RESPIRATION - ANTAGONIST PROFILE

被引:8
作者
RIBEIRO, JA
MONTEIRO, EC
机构
[1] Laboratory of Pharmacology, Gulbenkian Institute of Science, 2781 -, Oeiras
来源
NUCLEOSIDES & NUCLEOTIDES | 1991年 / 10卷 / 05期
关键词
D O I
10.1080/07328319108047232
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
The use of xanthines to characterize the adenosine receptor involved in excitation of respiration revealed that XCC, PD 115,199 and XAC have much higher affinities than DPCPX followed by PACPX, DPX and 8-PT, which is compatible with an A2 type of adenosine receptor.
引用
收藏
页码:945 / 953
页数:9
相关论文
共 16 条
[1]   PD 115,199 - AN ANTAGONIST LIGAND FOR ADENOSINE A2-RECEPTORS [J].
BRUNS, RF ;
FERGUS, JH ;
BADGER, EW ;
BRISTOL, JA ;
SANTAY, LA ;
HAYS, SJ .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 335 (01) :64-69
[2]   BINDING OF THE A1-SELECTIVE ADENOSINE ANTAGONIST 8-CYCLOPENTYL-1,3-DIPROPYLXANTHINE TO RAT-BRAIN MEMBRANES [J].
BRUNS, RF ;
FERGUS, JH ;
BADGER, EW ;
BRISTOL, JA ;
SANTAY, LA ;
HARTMAN, JD ;
HAYS, SJ ;
HUANG, CC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 335 (01) :59-63
[3]  
DALY JW, 1989, ADENOSINE RECEPTORS, P41
[4]  
DALY JW, 1987, TOPICS PERSPECTIVES, P23
[5]  
EVONIUK G, 1987, J PHARMACOL EXP THER, V242, P882
[6]   EVIDENCE THAT A NOVEL 8-PHENYL SUBSTITUTED XANTHINE DERIVATIVE IS A CARDIOSELECTIVE ADENOSINE RECEPTOR ANTAGONIST INVIVO [J].
FREDHOLM, BB ;
JACOBSON, KA ;
JONZON, B ;
KIRK, KL ;
LI, YO ;
DALY, JW .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1987, 9 (04) :396-400
[7]   8-SUBSTITUTED XANTHINES AS ANTAGONISTS AT A1-ADENOSINE AND A2-ADENOSINE RECEPTORS [J].
JACOBSON, KA ;
DELACRUZ, R ;
SCHULICK, R ;
KIRIASIS, L ;
PADGETT, W ;
PFLEIDERER, W ;
KIRK, KL ;
NEUMEYER, JL ;
DALY, JW .
BIOCHEMICAL PHARMACOLOGY, 1988, 37 (19) :3653-3661
[8]   8-CYCLOPENTYL-1,3-DIPROPYLXANTHINE (DPCPX) - A SELECTIVE HIGH-AFFINITY ANTAGONIST RADIOLIGAND FOR A1 ADENOSINE RECEPTORS [J].
LOHSE, MJ ;
KLOTZ, KN ;
LINDENBORNFOTINOS, J ;
REDDINGTON, M ;
SCHWABE, U ;
OLSSON, RA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 336 (02) :204-210
[9]   PHARMACOLOGICAL CHARACTERIZATION OF THE RECEPTOR INVOLVED IN CHEMOEXCITATION INDUCED BY ADENOSINE [J].
MCQUEEN, DS ;
RIBEIRO, JA .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 88 (03) :615-620
[10]  
MONTEIRO EC, 1987, N-S ARCH PHARMACOL, V335, P143