CYTIDINE AND DEOXYCYTIDYLATE DEAMINASE INHIBITION BY URIDINE ANALOGS

被引:24
作者
DRAKE, JC [1 ]
HANDE, KR [1 ]
FULLER, RW [1 ]
CHABNER, BA [1 ]
机构
[1] NCI,DIV CANC TREATMENT,PROGRAM DEV THERAPEUT,MED CHEM & BIOL LAB,BETHESDA,MD 20205
关键词
D O I
10.1016/0006-2952(80)90561-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:807 / 811
页数:5
相关论文
共 24 条
[1]   STUDIES OF ENZYMATIC DEAMINATION OF ARA-CYTIDINE .V. INHIBITION IN VITRO AND IN VIVO BY TETRAHYDROURIDINE AND OTHER REDUCED PYRIMIDINE NUCLEOSIDES [J].
CAMIENER, GW .
BIOCHEMICAL PHARMACOLOGY, 1968, 17 (09) :1981-&
[2]  
CAMIENER GW, 1967, BIOCH PHARMAC, V16, P1961
[3]   PURIFICATION AND PROPERTIES OF CYTIDINE DEAMINASE FROM NORMAL AND LEUKEMIC GRANULOCYTES [J].
CHABNER, BA ;
JOHNS, DG ;
COLEMAN, CN ;
DRAKE, JC ;
EVANS, WH .
JOURNAL OF CLINICAL INVESTIGATION, 1974, 53 (03) :922-931
[4]   CLINICAL PHARMACOLOGY OF ANTINEOPLASTIC AGENTS .1. [J].
CHABNER, BA ;
MYERS, CE ;
COLEMAN, N ;
JOHNS, DG .
NEW ENGLAND JOURNAL OF MEDICINE, 1975, 292 (21) :1107-1113
[5]  
CHANG P, 1977, P AM ASSOC CANC RES, V18, P352
[6]  
COLEMAN CN, 1975, BLOOD, V46, P791
[7]  
DAWSON WH, 1977, J CARB-NUCLEOS-NUCL, V4, P363
[8]  
HANDE KR, 1978, CANCER RES, V38, P597
[9]  
JACKSON RC, 1978, J BIOL CHEM, V253, P7440
[10]  
KREIS W, 1977, CANCER TREAT REP, V61, P1347