STUDIES IN INDOLE SERIES .4. TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLES AS SEROTONIN ANTAGONISTS

被引：17

作者：

CATTANACH, CJ

COHEN, A

HEATHBRO.B

机构：

[1] Roche Products Ltd., Welwyn Garden City, Herts., Broadwater Road

来源：

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC | 1968年 / 10期

关键词：

D O I：

10.1039/j39680001235

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of tetrahydro-1H-pyrido [4,3-b] indoles has been made by Fischer cyclisation of arylhydrazones of 1-substituted-4-piperidones. Some of these compounds have been shown to have high anti-serotonin activity when submitted to pharmocological tests in vitro.

引用

页码：1235 / +

页数：1

共 33 条

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