SYNTHESIS OF THE BETA-LACTONE ESTERASE INHIBITOR VALILACTONE USING PI-ALLYLTRICARBONYLIRON LACTONE COMPLEXES

被引：33

作者：

BATES, RW ^{[1
]}

FERNANDEZMORO, R ^{[1
]}

LEY, SV ^{[1
]}

机构：

[1] IMPERIAL COLL SCI TECHNOL & MED,DEPT CHEM,LONDON SW7 2AY,ENGLAND

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 23期

关键词：

D O I：

10.1016/S0040-4039(00)78809-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of the esterase inhibitor valilactone (1) is reported employing the oxidation of pi-allyltricarbonyliron lactone complexes with ceric ammonium nitrate to afford the inherent beta-lactone ring.

引用

页码：2651 / 2654

页数：4

共 24 条

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