SYNTHESIS AND TUMOR UPTAKE OF 5-HALO-1-(2'-FLUORO-2'-DEOXY-BETA-D-RIBOFURANOSYL)[2-C-14]URACILS

被引：30

作者：

MERCER, JR ^{[1
]}

KNAUS, EE ^{[1
]}

WIEBE, LI ^{[1
]}

机构：

[1] UNIV ALBERTA,FAC PHARM & PHARMACEUT SCI,EDMONTON T6G 2N8,ALBERTA,CANADA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 04期

关键词：

D O I：

10.1021/jm00387a015

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：670 / 675

页数：6

共 31 条

[1] STUDIES ON F-18-LABELED PYRIMIDINES - TUMOR UPTAKES OF 5-FLUOROURACIL-F-18, 5-FLUOROURIDINE-F-18, AND 5-FLUORODEOXYURIDINE-F-18 IN ANIMALS [J].

ABE, Y ;

FUKUDA, H ;

ISHIWATA, K ;

YOSHIOKA, S ;

YAMADA, K ;

ENDO, S ;

KUBOTA, K ;

SATO, T ;

MATSUZAWA, T ;

TAKAHASHI, T ;

IDO, T .

EUROPEAN JOURNAL OF NUCLEAR MEDICINE, 1983, 8 (06) :258-261

[2] TUMOR UPTAKE OF RADIOLABELED PYRIMIDINE-BASES AND PYRIMIDINE NUCLEOSIDES IN ANIMAL-MODELS .1. 5-FLUOROURACIL-6-H-3 [J].

ABRAMS, DN ;

KNAUS, EE ;

WIEBE, LI .

INTERNATIONAL JOURNAL OF NUCLEAR MEDICINE & BIOLOGY, 1979, 6 (02) :97-101

[3] THE SYNTHESIS OF RADIOLABELED 1-(2'-FLUORO-2'-DEOXY-BETA-D-RIBOFURANOSYL)URACIL AND 1-(2'-CHLORO-2'-DEOXY-BETA-D-RIBOFURANOSYL)URACIL [J].

ABRAMS, DN ;

MERCER, JR ;

KNAUS, EE ;

WIEBE, LI .

INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES, 1985, 36 (03) :233-238

[4]

ABRAMS DN, 1978, CHEM RADIOPHARMACEUT, P205

[5]

ABRAMS DN, 1985, BRIT J RADIOL, V59, P263

[6] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 5-FLUORO-2',3'-DIDEOXY-3'-FLUOROURIDINE AND ITS 5'-PHOSPHATE [J].

AJMERA, S ;

BAPAT, AR ;

DANENBERG, K ;

DANENBERG, PV .

JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (01) :11-14

[7] EFFECTS OF 5-TRIFLUOROMETHYLDEOXYURIDINE UPON DEOXYTHYMIDINE KINASE [J].

BRESNICK, E ;

WILLIAMS, SS .

BIOCHEMICAL PHARMACOLOGY, 1967, 16 (03) :503-&

[8] NUCLEIC-ACID COMPONENTS AND THEIR ANALOGS .186. PREPARATION OF SOME 2'-DEOXY-5-FLUOROURIDINE DERIVATIVES BY A DIRECT FLUORINATION [J].

CECH, D ;

HOLY, A .

COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1976, 41 (11) :3335-3342

[9]

CODERRE JA, 1983, J MED CHEM, V26, P1149

[10] NUCLEOSIDES .14. SYNTHESIS OF 2'-DEOXY-2'-FLUOROURIDINE [J].

CODINGTON, JF ;

FOX, JJ ;

VANPRAAG, D ;

BENDICH, A ;

DOERR, I .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1961, 83 (24) :5030-+

← 1 2 3 4 →