CEREBROVASODILATATION THROUGH SELECTIVE-INHIBITION OF THE ENZYME CARBONIC-ANHYDRASE .3. 5-(ARYLTHIO)-, 5-(ARYLSULFINYL)-, AND 5-(ARYLSULFONYL)THIOPHENE-2-SULFONAMIDES

被引：16

作者：

BARNISH, IT ^{[1
]}

CROSS, PE ^{[1
]}

DICKINSON, RP ^{[1
]}

PARRY, MJ ^{[1
]}

RANDALL, MJ ^{[1
]}

机构：

[1] PFIZER LTD,PFIZER CENT RES,SANDWICH,KENT,ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 08期

关键词：

D O I：

10.1021/jm00140a009

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：959 / 964

页数：6

共 18 条

[1] CEREBROVASODILATATION THROUGH SELECTIVE-INHIBITION OF THE ENZYME CARBONIC-ANHYDRASE .2. IMIDAZO[2,1-B]THIADIAZOLE AND IMIDAZO[2,1-B]THIAZOLESULFONAMIDES [J].

BARNISH, IT ;

CROSS, PE ;

DICKINSON, RP ;

GADSBY, B ;

PARRY, MJ ;

RANDALL, MJ ;

SINCLAIR, IW .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (02) :117-121

[2]

BUZAS A, 1961, ANN PHARM FR, V19, P449

[3] CEREBRO-VASODILATATION THROUGH SELECTIVE-INHIBITION OF ENZYME CARBONIC-ANHYDRASE .1. SUBSTITUTED BENZENEDISULFONAMIDES [J].

CROSS, PE ;

GADSBY, B ;

HOLLAND, GF ;

MCLAMORE, WM .

JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (09) :845-850

[4] INFLUENCE OF ACETAZOLAMIDE ON CEREBRAL BLOOD FLOW [J].

EHRENREICH, D ;

BURNS, RA ;

FAZEKAS, JF ;

ALMAN, RW .

ARCHIVES OF NEUROLOGY, 1961, 5 (02) :227-&

[5] CARBONIC ANHYDRASE INHIBITION AND CEREBRAL VENOUS BLOOD GASES AND IONS IN MAN - DEMONSTRATION OF INCREASED OXYGEN AVAILABILITY TO ISCHEMIC BRAIN [J].

GOTOH, F ;

MEYER, JS ;

TOMITA, M .

ARCHIVES OF INTERNAL MEDICINE, 1966, 117 (01) :39-+

[6]

GRAY WD, 1967, J PHARMACOL EXP THER, V156, P383

[7]

GRAY WD, 1957, J PHARMACOL EXP THER, V121, P160

[8]

HARPER AM, 1965, ACTA NEUROL SCAND S, V14, P94

[9]

HO TL, 1972, SYNTHESIS, V10, P561

[10]

KAKEYA F, 1969, CHEM PHARM B, V17, P2000

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